Design, synthesis, and biological evaluation of a new class of small molecule peptide mimetics targeting the melanocortin receptors.
about
Design, synthesis and biological evaluation of ligands selective for the melanocortin-3 receptorStructure-activity relationships of cyclic lactam analogues of alpha-melanocyte-stimulating hormone (alpha-MSH) targeting the human melanocortin-3 receptorDesign of novel melanocortin receptor ligands: multiple receptors, complex pharmacology, the challengeSolid-phase peptide head-to-side chain cyclodimerization: discovery of C(2)-symmetric cyclic lactam hybrid α-melanocyte-stimulating hormone (MSH)/agouti-signaling protein (ASIP) analogues with potent activities at the human melanocortin receptorsMelanotropins as drugs for the treatment of obesity and other feeding disorders: potential and problems.Approaches to the rational design of selective melanocortin receptor antagonists.Design of peptide and peptidomimetic ligands with novel pharmacological activity profiles.Substitution of arginine with proline and proline derivatives in melanocyte-stimulating hormones leads to selectivity for human melanocortin 4 receptor.Adventures in peptides and science with students! The joys of research.The first preparative solution phase synthesis of melanotan II.Beta-turn secondary structure and melanocortin ligands.
P2860
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P2860
Design, synthesis, and biological evaluation of a new class of small molecule peptide mimetics targeting the melanocortin receptors.
description
2006 nî lūn-bûn
@nan
2006年の論文
@ja
2006年論文
@yue
2006年論文
@zh-hant
2006年論文
@zh-hk
2006年論文
@zh-mo
2006年論文
@zh-tw
2006年论文
@wuu
2006年论文
@zh
2006年论文
@zh-cn
name
Design, synthesis, and biologi ...... ng the melanocortin receptors.
@en
type
label
Design, synthesis, and biologi ...... ng the melanocortin receptors.
@en
prefLabel
Design, synthesis, and biologi ...... ng the melanocortin receptors.
@en
P2093
P2860
P1476
Design, synthesis, and biologi ...... ng the melanocortin receptors.
@en
P2093
Alexander V Mayorov
Dev Trivedi
James P Cain
Minying Cai
Ravil R Petrov
Victor J Hruby
YeonSun Lee
P2860
P304
P356
10.1016/J.BMCL.2006.07.015
P407
P577
2006-08-22T00:00:00Z