Low affinity analogs of thyrotropin-releasing hormone are super-agonists. - Test2 - elhamkhani - TriplyDB

Low affinity analogs of thyrotropin-releasing hormone are super-agonists.

Low affinity analogs of thyrotropin-releasing hormone are super-agonists.

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Hypothalamic neurohormones and immune responses.A novel TRH analog, Glp-Asn-Pro-D-Tyr-D-TrpNH2, binds to [3H][3-Me-His2]TRH-labelled sites in rat hippocampus and cortex but not pituitary or heterologous cells expressing TRHR1 or TRHR2.Thyrotropin receptor stimulates internalization-independent persistent phosphoinositide signaling Discovery of a low affinity thyrotropin-releasing hormone (TRH)-like peptide that exhibits potent inhibition of scopolamine-induced memory impairment in mice.Taltirelin is a superagonist at the human thyrotropin-releasing hormone receptor Synthesis, receptor binding, and CNS pharmacological studies of new thyrotropin-releasing hormone (TRH) analogues.Thyrotropin-releasing hormone receptor type 1 (TRH-R1), not TRH-R2, primarily mediates taltirelin actions in the CNS of mice.Discovery of novel agonists and antagonists of the free fatty acid receptor 1 (FFAR1) using virtual screening.Novel thyrotropin-releasing hormone analogs: a patent review.Superagonism at G protein-coupled receptors and beyond.Long Receptor Residence Time of C26 Contributes to Super Agonist Activity at the Human β2 Adrenoceptor.Functional characterization of human bitter taste receptors.

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P2860

Low affinity analogs of thyrotropin-releasing hormone are super-agonists.

http://www.wikidata.org/entity/Q40301576

description

2006 nî lūn-bûn

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2006年の論文

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2006年論文

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2006年論文

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2006年論文

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2006年論文

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2006年論文

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2006年论文

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2006年论文

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2006年论文

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name

Low affinity analogs of thyrotropin-releasing hormone are super-agonists.

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type

label

Low affinity analogs of thyrotropin-releasing hormone are super-agonists.

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prefLabel

Low affinity analogs of thyrotropin-releasing hormone are super-agonists.

@en

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P1433

Journal of Biological Chemistry

P1476

Low affinity analogs of thyrotropin-releasing hormone are super-agonists.

@en

P2093

John Northup

http://www.w3.org/2001/XMLSchema#string

Marvin C Gershengorn

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Navneet Kaur

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Rahul Jain

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Stanislav Engel

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Susanne Neumann

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Vikramdeep Monga

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P2860

G protein-coupled receptors: a count of 1001 conformations

Concanamycin A, the specific inhibitor of V-ATPases, binds to the V(o) subunit c.

Static and dynamic roles of extracellular loops in G-protein-coupled receptors: a mechanism for sequential binding of thyrotropin-releasing hormone to its receptor.

Thyrotropin-releasing hormone receptors -- similarities and differences.

The novel and specific Rho-kinase inhibitor (S)-(+)-2-methyl-1-[(4-methyl-5-isoquinoline)sulfonyl]-homopiperazine as a probing molecule for Rho-kinase-involved pathway.

Regulation of G protein-coupled receptor kinases and arrestins during receptor desensitization.

Ligand-selective receptor conformations revisited: the promise and the problem.

Prenyl modification of guanine nucleotide regulatory protein gamma 2 subunits is not required for interaction with the transducin alpha subunit or rhodopsin

Mechanism of signal transduction by TRH.

Kinetic analysis of the internalization and recycling of [3H]TRH and C-terminal truncations of the long isoform of the rat thyrotropin-releasing hormone receptor-1.

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13103-13109

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scholarly article

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10.1074/JBC.M600440200

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19

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281

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2006-03-21T00:00:00Z

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16551618

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