Peripheral 5-HT2-like receptors. Can they be classified with the available antagonists?
about
Long-lasting target binding and rebinding as mechanisms to prolong in vivo drug actionActivation of meningeal 5-HT2B receptors: an early step in the generation of migraine headache?GR32191, a highly potent and specific thromboxane A2 receptor blocking drug on platelets and vascular and airways smooth muscle in vitroThe classification of peripheral 5-HT2-like receptors using tryptamine agonist and antagonist analoguesNew insights in insurmountable antagonism.Classification of platelet and vascular prostaglandin D2 (DP) receptors: estimation of affinities and relative efficacies for a series of novel bicyclic ligands. With an appendix on goodness-of-fit analyses.Heterogeneity of thromboxane A2 (TP-) receptors: evidence from antagonist but not agonist potency measurements.Elusive equilibrium: the challenge of interpreting receptor pharmacology using calcium assays.Clozapine, atypical antipsychotics, and the benefits of fast-off D2 dopamine receptor antagonism.The classification of 5-hydroxytryptamine receptors.On the different experimental manifestations of two-state 'induced-fit' binding of drugs to their cellular targetsThe classification of 5-hydroxytryptamine receptors.The role of serotonin in schizophrenia: an overview of the nomenclature, distribution and alterations of serotonin receptors in the central nervous system.Differential classification of vascular smooth muscle and endothelial cell 5-HT receptors by use of tryptamine analogues.Analysis of the agonist activity of fenoldopam (SKF 82526) at the vascular 5-HT2 receptor.Involvement of 5-HT(1B/1D) and 5-HT2A receptors in 5-HT-induced contraction of endothelium-denuded rabbit epicardial coronary arteries.5-hydroxytryptamine receptors mediating vasoconstriction and vasodilation in perinatal and adult rabbit small pulmonary arteries.Actions of non-peptide ergot alkaloids at 5-HT1-like and 5-HT2 receptors mediating vascular smooth muscle contraction.Differences in agonist dissociation constant estimates for 5-HT at 5-HT2-receptors: a problem of acute desensitization?Effect of the thromboxane A2-mimetic U46619 on 5-HT1-like and 5-HT2 receptor-mediated contraction of the rabbit isolated femoral artery.Analysis of the effects of alpha 1-adrenoceptor antagonists on noradrenaline-mediated contraction of rat small mesenteric arteryInvolvement of 5-HT1B receptors in collar-induced hypersensitivity to 5-hydroxytryptamine of the rabbit carotid artery.Analysis of the 5-HT receptor in rabbit saphenous vein exemplifies the problems of using exclusion criteria for receptor classification.Comparative analysis of two types of 5-hydroxytryptamine receptor mediating vasorelaxation: differential classification using tryptamines.
P2860
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P2860
Peripheral 5-HT2-like receptors. Can they be classified with the available antagonists?
description
1986 nî lūn-bûn
@nan
1986年の論文
@ja
1986年論文
@yue
1986年論文
@zh-hant
1986年論文
@zh-hk
1986年論文
@zh-mo
1986年論文
@zh-tw
1986年论文
@wuu
1986年论文
@zh
1986年论文
@zh-cn
name
Peripheral 5-HT2-like receptors. Can they be classified with the available antagonists?
@en
Peripheral 5-HT2-like receptors. Can they be classified with the available antagonists?
@nl
type
label
Peripheral 5-HT2-like receptors. Can they be classified with the available antagonists?
@en
Peripheral 5-HT2-like receptors. Can they be classified with the available antagonists?
@nl
prefLabel
Peripheral 5-HT2-like receptors. Can they be classified with the available antagonists?
@en
Peripheral 5-HT2-like receptors. Can they be classified with the available antagonists?
@nl
P2860
P1476
Peripheral 5-HT2-like receptors. Can they be classified with the available antagonists?
@en
P2093
P2860
P304
P356
10.1111/J.1476-5381.1986.TB10239.X
P407
P577
1986-07-01T00:00:00Z