BAY60-6583 acts as a partial agonist at adenosine A2B receptors.
about
Probing biased/partial agonism at the G protein-coupled A(2B) adenosine receptor.Medicinal chemistry of adenosine, P2Y and P2X receptors.A Novel Method for Screening Adenosine Receptor Specific Agonists for Use in Adenosine Drug Development.Selectivity is species-dependent: Characterization of standard agonists and antagonists at human, rat, and mouse adenosine receptors.On the G protein-coupling selectivity of the native A2B adenosine receptor.Characterisation of endogenous A2A and A2B receptor-mediated cyclic AMP responses in HEK 293 cells using the GloSensor™ biosensor: Evidence for an allosteric mechanism of action for the A2B-selective antagonist PSB 603.Adenosine A2A receptor ligand recognition and signaling is blocked by A2B receptors.
P2860
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P2860
BAY60-6583 acts as a partial agonist at adenosine A2B receptors.
description
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name
BAY60-6583 acts as a partial agonist at adenosine A2B receptors.
@en
BAY60-6583 acts as a partial agonist at adenosine A2B receptors.
@nl
type
label
BAY60-6583 acts as a partial agonist at adenosine A2B receptors.
@en
BAY60-6583 acts as a partial agonist at adenosine A2B receptors.
@nl
prefLabel
BAY60-6583 acts as a partial agonist at adenosine A2B receptors.
@en
BAY60-6583 acts as a partial agonist at adenosine A2B receptors.
@nl
P2093
P356
P1476
BAY60-6583 acts as a partial agonist at adenosine A2B receptors.
@en
P2093
Benjamin F Seibt
Sonja Hinz
Svenja K Lacher
P304
P356
10.1124/JPET.113.210849
P407
P577
2014-03-14T00:00:00Z