Highly potent and selective fluorescent antagonists of the human adenosine A₃ receptor based on the 1,2,4-triazolo[4,3-a]quinoxalin-1-one scaffold.
about
Fluorescent approaches for understanding interactions of ligands with G protein coupled receptorsApplication of BRET to monitor ligand binding to GPCRs.Fluorescent ligands for adenosine receptors.Characterization by flow cytometry of fluorescent, selective agonist probes of the A(3) adenosine receptor.Biophysical Detection of Diversity and Bias in GPCR Function.High-Affinity Functional Fluorescent Ligands for Human β-Adrenoceptors.Detection of the secondary, low-affinity β1 -adrenoceptor site in living cells using the fluorescent CGP 12177 derivative BODIPY-TMR-CGP.Synthesis of BODIPY derivatives substituted with various bioconjugatable linker groups: a construction kit for fluorescent labeling of receptor ligands.Development of novel fluorescent histamine H1-receptor antagonists to study ligand-binding kinetics in living cells.A Non-imaging High Throughput Approach to Chemical Library Screening at the Unmodified Adenosine-A3 Receptor in Living Cells.Nanomolar-Potency 1,2,4-Triazoloquinoxaline Inhibitors of the Kidney Urea Transporter UT-A1.
P2860
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P2860
Highly potent and selective fluorescent antagonists of the human adenosine A₃ receptor based on the 1,2,4-triazolo[4,3-a]quinoxalin-1-one scaffold.
description
2012 nî lūn-bûn
@nan
2012年の論文
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2012年学术文章
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2012年学术文章
@zh
2012年学术文章
@zh-cn
2012年学术文章
@zh-hans
2012年学术文章
@zh-my
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2012年學術文章
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2012年學術文章
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name
Highly potent and selective fl ...... 3-a]quinoxalin-1-one scaffold.
@en
Highly potent and selective fl ...... 3-a]quinoxalin-1-one scaffold.
@nl
type
label
Highly potent and selective fl ...... 3-a]quinoxalin-1-one scaffold.
@en
Highly potent and selective fl ...... 3-a]quinoxalin-1-one scaffold.
@nl
prefLabel
Highly potent and selective fl ...... 3-a]quinoxalin-1-one scaffold.
@en
Highly potent and selective fl ...... 3-a]quinoxalin-1-one scaffold.
@nl
P50
P356
P1476
Highly potent and selective fl ...... ,3-a]quinoxalin-1-one scaffold
@en
P2093
Barrie Kellam
P304
P356
10.1021/JM201722Y
P407
P577
2012-02-13T00:00:00Z