about
Kinetic target-guided synthesis in drug discovery and chemical biology: a comprehensive facts and figures surveyComparative Study of the Synthesis and Structural and Physicochemical Properties of Diketopiperazines vs Aza-diketopiperazines.Discovery of a new class of protein farnesyltransferase inhibitors in the arylthiophene series.Structure-activity relationships of imidazole-derived 2-[N-carbamoylmethyl-alkylamino]acetic acids, dual binders of human insulin-degrading enzyme.Highly improved antiparasitic activity after introduction of an N-benzylimidazole moiety on protein farnesyltransferase inhibitors.Catalytic site inhibition of insulin-degrading enzyme by a small molecule induces glucose intolerance in micePrecision autophagy: Will the next wave of selective autophagy markers and specific autophagy inhibitors feed clinical pipelines?Aggrecanase-2 inhibitors based on the acylthiosemicarbazide zinc-binding group.Development of fluorescent peptide substrates and assays for the key autophagy-initiating cysteine protease enzyme, ATG4B.New protein farnesyltransferase inhibitors in the 3-arylthiophene 2-carboxylic acid series: diversification of the aryl moiety by solid-phase synthesis.Controlling Plasma Stability of Hydroxamic Acids: A MedChem Toolbox.A new quinoline-based chemical probe inhibits the autophagy-related cysteine protease ATG4BIdentification of ebselen as a potent inhibitor of insulin degrading enzyme by a drug repurposing screeningKinetic Target-Guided Synthesis: Reaching the Age of Maturity
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description
researcher
@en
wetenschapper
@nl
հետազոտող
@hy
name
Damien Bosc
@ast
Damien Bosc
@en
Damien Bosc
@es
Damien Bosc
@nl
type
label
Damien Bosc
@ast
Damien Bosc
@en
Damien Bosc
@es
Damien Bosc
@nl
prefLabel
Damien Bosc
@ast
Damien Bosc
@en
Damien Bosc
@es
Damien Bosc
@nl
P108
P106
P108
P1153
40260955300
P31
P496
0000-0002-6076-2934