HU-243
HU-243 (AM-4056) is a synthetic cannabinoid drug that is a single enantiomer of the hydrogenated derivative of the commonly used reference agonist HU-210. It is a potent agonist at both the CB1 and CB2 receptors, with a binding affinity of 0.041 nM at the CB1 receptor, making it marginally more potent than HU-210, which had an affinity of 0.061 nM in the same assay.
primaryTopic
HU-243
HU-243 (AM-4056) is a synthetic cannabinoid drug that is a single enantiomer of the hydrogenated derivative of the commonly used reference agonist HU-210. It is a potent agonist at both the CB1 and CB2 receptors, with a binding affinity of 0.041 nM at the CB1 receptor, making it marginally more potent than HU-210, which had an affinity of 0.061 nM in the same assay.
has abstract
HU-243 (AM-4056) is a syntheti ...... of 0.061 nM in the same assay.
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CAS number
140835-18-3
IUPAC name
(6aR,8S,9S,10aR)-9-(hydroxymet ...... hydro-6aH-benzo[c]chromen-1-ol
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PubChem
Wikipage page ID
28,806,935
Wikipage revision ID
732,523,719
IUPHAR ligand
molecular weight
smiles
CC[C@H]2[C@@H]C3=C1C=CC=C3O
comment
HU-243 (AM-4056) is a syntheti ...... of 0.061 nM in the same assay.
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label
HU-243
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