ZK-93426
ZK-93426 (ethyl-5-isopropoxy-4-methyl-beta-carboline-3-carboxylate) is a drug from the beta-carboline family. It acts as a weak partial inverse agonist of benzodiazepine receptors, meaning that it causes the opposite effects to the benzodiazepine class of drugs and has anxiogenic properties, although unlike most benzodiazepine antagonists it is not a convulsant and actually has weak anticonvulsant effects. In human tests it produced alertness, restlessness and feelings of apprehension, and reversed the effect of the benzodiazepine lormetazepam. It was also shown to produce nootropic effects and increased release of acetylcholine.
primaryTopic
ZK-93426
ZK-93426 (ethyl-5-isopropoxy-4-methyl-beta-carboline-3-carboxylate) is a drug from the beta-carboline family. It acts as a weak partial inverse agonist of benzodiazepine receptors, meaning that it causes the opposite effects to the benzodiazepine class of drugs and has anxiogenic properties, although unlike most benzodiazepine antagonists it is not a convulsant and actually has weak anticonvulsant effects. In human tests it produced alertness, restlessness and feelings of apprehension, and reversed the effect of the benzodiazepine lormetazepam. It was also shown to produce nootropic effects and increased release of acetylcholine.
has abstract
ZK-93426 (ethyl-5-isopropoxy-4 ...... ased release of acetylcholine.
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IUPAC name
ethyl 5-​isopropoxy-&#x ...... -​3-​carboxylate
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thumbnail
Wikipage page ID
20,107,077
Wikipage revision ID
670,406,335
othernames
ZK-93426; ethyl 4-methyl-5-propan-2-yloxy-9H-pyrido[5,4-b]indole-3-carboxylate
Verifiedfields
verifiedrevid
445,991,871
Watchedfields
subject
comment
ZK-93426 (ethyl-5-isopropoxy-4 ...... ased release of acetylcholine.
@en
label
ZK-93426
@en