EDG6, a novel G-protein-coupled receptor related to receptors for bioactive lysophospholipids, is specifically expressed in lymphoid tissue
about
Discovery, design and synthesis of novel potent and selective sphingosine-1-phosphate 4 receptor (S1P₄-R) agonistsEdg-1, the G protein-coupled receptor for sphingosine-1-phosphate, is essential for vascular maturationDifferential pharmacological properties and signal transduction of the sphingosine 1-phosphate receptors EDG-1, EDG-3, and EDG-5Nrg-1 belongs to the endothelial differentiation gene family of G protein-coupled sphingosine-1-phosphate receptorsTandem genomic arrangement of a G protein (Gna15) and G protein-coupled receptor (s1p(4)/lp(C1)/Edg6) geneInhibitory regulation of Rac activation, membrane ruffling, and cell migration by the G protein-coupled sphingosine-1-phosphate receptor EDG5 but not EDG1 or EDG3Sphingosine 1-Phosphate Receptors: Do They Have a Therapeutic Potential in Cardiac Fibrosis?Discovery, design and synthesis of the first reported potent and selective sphingosine-1-phosphate 4 (S1P4) receptor antagonists.An update on the biology of sphingosine 1-phosphate receptors.Sphingosine 1-phosphate signalling in mammalian cells.The sphingosine 1-phosphate transporter, SPNS2, functions as a transporter of the phosphorylated form of the immunomodulating agent FTY720.Extracellular and intracellular actions of sphingosine-1-phosphateSystemic distribution, subcellular localization and differential expression of sphingosine-1-phosphate receptors in benign and malignant human tissues.Sphingosine 1-phosphate receptor 4 uses HER2 (ERBB2) to regulate extracellular signal regulated kinase-1/2 in MDA-MB-453 breast cancer cellsModulation of chemokines and allergic airway inflammation by selective local sphingosine-1-phosphate receptor 1 agonism in lungs"Inside-out" signaling of sphingosine-1-phosphate: therapeutic targets.Sphingosine-1-phosphate lyase deficiency produces a pro-inflammatory response while impairing neutrophil trafficking.Discovery, design and synthesis of a selective S1P(3) receptor allosteric agonist.Cardiovascular effects of sphingosine-1-phosphate and other sphingomyelin metabolites.S1P is associated with protection in human and experimental cerebral malariaSphingosine-1-phosphate receptor 2CFTR and sphingolipids mediate hypoxic pulmonary vasoconstrictionRegulation of mammalian physiology, development, and disease by the sphingosine 1-phosphate and lysophosphatidic acid receptors.Insights into the pharmacological relevance of lysophospholipid receptors.Roles of sphingosine-1-phosphate (S1P) receptors in malignant behavior of glioma cells. Differential effects of S1P2 on cell migration and invasiveness.The role of sphingosine-1-phosphate in breast cancer tumor-induced lymphangiogenesis.Sphingolipids and membrane biology as determined from genetic models.Sphingosine 1-phosphate receptor signaling regulates proper embryonic vascular patterning.G protein-coupled receptors as therapeutic targets for multiple sclerosis.Cardioprotection in ischemia/reperfusion injury: spotlight on sphingosine-1-phosphate and bradykinin signalling.Sphingosine 1-phosphate in coagulation and inflammation.Beyond Immune Cell Migration: The Emerging Role of the Sphingosine-1-phosphate Receptor S1PR4 as a Modulator of Innate Immune Cell Activation.Clinical pharmacology, efficacy, and safety aspects of sphingosine-1-phosphate receptor modulators.Targeting sphingosine-1-phosphate signaling for cancer therapy.S1P(4) receptor mediates S1P-induced vasoconstriction in normotensive and hypertensive rat lungs.S1P(5) is required for sphingosine 1-phosphate-induced autophagy in human prostate cancer PC-3 cells.Lysophospholipid signaling: beyond the EDGs.Sphingosine 1-phosphate analogue recognition and selectivity at S1P4 within the endothelial differentiation gene family of receptors.Pharmacological characterization of human S1P4 using a novel radioligand, [4,5-3H]-dihydrosphingosine-1-phosphate.G-protein-coupled receptor stimulation of the p42/p44 mitogen-activated protein kinase pathway is attenuated by lipid phosphate phosphatases 1, 1a, and 2 in human embryonic kidney 293 cells.
P2860
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P2860
EDG6, a novel G-protein-coupled receptor related to receptors for bioactive lysophospholipids, is specifically expressed in lymphoid tissue
description
1998 nî lūn-bûn
@nan
1998 թուականի Հոկտեմբերին հրատարակուած գիտական յօդուած
@hyw
1998 թվականի հոտեմբերին հրատարակված գիտական հոդված
@hy
1998年の論文
@ja
1998年論文
@yue
1998年論文
@zh-hant
1998年論文
@zh-hk
1998年論文
@zh-mo
1998年論文
@zh-tw
1998年论文
@wuu
name
EDG6, a novel G-protein-couple ...... y expressed in lymphoid tissue
@ast
EDG6, a novel G-protein-couple ...... y expressed in lymphoid tissue
@en
EDG6, a novel G-protein-couple ...... y expressed in lymphoid tissue
@en-gb
EDG6, a novel G-protein-couple ...... y expressed in lymphoid tissue
@nl
type
label
EDG6, a novel G-protein-couple ...... y expressed in lymphoid tissue
@ast
EDG6, a novel G-protein-couple ...... y expressed in lymphoid tissue
@en
EDG6, a novel G-protein-couple ...... y expressed in lymphoid tissue
@en-gb
EDG6, a novel G-protein-couple ...... y expressed in lymphoid tissue
@nl
prefLabel
EDG6, a novel G-protein-couple ...... y expressed in lymphoid tissue
@ast
EDG6, a novel G-protein-couple ...... y expressed in lymphoid tissue
@en
EDG6, a novel G-protein-couple ...... y expressed in lymphoid tissue
@en-gb
EDG6, a novel G-protein-couple ...... y expressed in lymphoid tissue
@nl
P921
P356
P1433
P1476
EDG6, a novel G-protein-couple ...... y expressed in lymphoid tissue
@en
P2093
P304
P356
10.1006/GENO.1998.5491
P407
P577
1998-10-01T00:00:00Z