N[3-(4'-fluorophenyl)-3-(4'-phenylphenoxy)propyl]sarcosine (NFPS) is a selective persistent inhibitor of glycine transport
about
Glycine transport inhibitors for the treatment of schizophreniaMolecular targets for treating cognitive dysfunction in schizophrenia.Dynamics of forward and reverse transport by the glial glycine transporter, glyt1b.N-arachidonyl-glycine modulates synaptic transmission in superficial dorsal hornGlutamatergic targets for enhancing extinction learning in drug addictionWhy glycine transporters have different stoichiometries.The therapeutic potential of glycine transporter-1 inhibitors.Targeting prefrontal cortical dopamine D1 and N-methyl-D-aspartate receptor interactions in schizophrenia treatment.Oleoyl-L-carnitine inhibits glycine transport by GlyT2Recent advances in the development of novel pharmacological agents for the treatment of cognitive impairments in schizophrenia.Synaptic homeostasis in a zebrafish glial glycine transporter mutant.Validation of a fluorescent imaging plate reader membrane potential assay for high-throughput screening of glycine transporter modulators.Glycine transport accounts for the differential role of glycine vs. D-serine at NMDA receptor coagonist sites in the salamander retina.The glycine transporter GlyT1 controls N-methyl-D-aspartic acid receptor coagonist occupancy in the mouse retina.Arachidonic acid and anandamide have opposite modulatory actions at the glycine transporter, GLYT1a.Glycine tranporter-1 blockade potentiates NMDA-mediated responses in rat prefrontal cortical neurons in vitro and in vivo.Blockade of glycine transporter-1 (GLYT-1) potentiates NMDA receptor-mediated synaptic transmission in hypoglossal motorneurons.Bergmann glial GlyT1 mediates glycine uptake and release in mouse cerebellar slices.The glycine transport inhibitor sarcosine is an NMDA receptor co-agonist that differs from glycine.Neurochemical, electrophysiological and pharmacological profiles of the selective inhibitor of the glycine transporter-1 SSR504734, a potential new type of antipsychotic.Molecular basis for substrate discrimination by glycine transporters.Glycine release provoked by disturbed Na⁺, Na⁺ and Ca²⁺ homeostasis in cerebellar nerve endings: roles of Ca²⁺ channels, Na⁺/Ca²⁺ exchangers and GlyT2 transporter reversal.
P2860
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P2860
N[3-(4'-fluorophenyl)-3-(4'-phenylphenoxy)propyl]sarcosine (NFPS) is a selective persistent inhibitor of glycine transport
description
2001 nî lūn-bûn
@nan
2001 թուականի Դեկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2001 թվականի դեկտեմբերին հրատարակված գիտական հոդված
@hy
2001年の論文
@ja
2001年論文
@yue
2001年論文
@zh-hant
2001年論文
@zh-hk
2001年論文
@zh-mo
2001年論文
@zh-tw
2001年论文
@wuu
name
N[3-(4'-fluorophenyl)-3-(4'-ph ...... inhibitor of glycine transport
@ast
N[3-(4'-fluorophenyl)-3-(4'-ph ...... inhibitor of glycine transport
@en
N[3-(4'-fluorophenyl)-3-(4'-ph ...... inhibitor of glycine transport
@nl
type
label
N[3-(4'-fluorophenyl)-3-(4'-ph ...... inhibitor of glycine transport
@ast
N[3-(4'-fluorophenyl)-3-(4'-ph ...... inhibitor of glycine transport
@en
N[3-(4'-fluorophenyl)-3-(4'-ph ...... inhibitor of glycine transport
@nl
prefLabel
N[3-(4'-fluorophenyl)-3-(4'-ph ...... inhibitor of glycine transport
@ast
N[3-(4'-fluorophenyl)-3-(4'-ph ...... inhibitor of glycine transport
@en
N[3-(4'-fluorophenyl)-3-(4'-ph ...... inhibitor of glycine transport
@nl
P2860
P356
P1476
N[3-(4'-fluorophenyl)-3-(4'-ph ...... inhibitor of glycine transport
@en
P2093
K R Aubrey
R J Vandenberg
P2860
P304
P356
10.1038/SJ.BJP.0704381
P407
P577
2001-12-01T00:00:00Z