A single histidine in GABAA receptors is essential for benzodiazepine agonist binding
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Ethanol potently and competitively inhibits binding of the alcohol antagonist Ro15-4513 to alpha4/6beta3delta GABAA receptorsDiazepam-bound GABAA receptor models identify new benzodiazepine binding-site ligandsUnravelling the mechanism of action of NS9283, a positive allosteric modulator of (α4)3(β2)2 nicotinic ACh receptorsAbuse and dependence liability of benzodiazepine-type drugs: GABA(A) receptor modulation and beyondPharmacological characterization of a novel cell line expressing human alpha(4)beta(3)delta GABA(A) receptorsSelective labelling of diazepam-insensitive GABAA receptors in vivo using [3H]Ro 15-4513Pentameric ligand-gated ion channel ELIC is activated by GABA and modulated by benzodiazepinesPrinciples of agonist recognition in Cys-loop receptorsAnxioselective anxiolytics: on a quest for the Holy GrailRole of the histidine residue at position 105 in the human alpha 5 containing GABA(A) receptor on the affinity and efficacy of benzodiazepine site ligandsAlterations in brain-derived neurotrophic factor in the mouse hippocampus following acute but not repeated benzodiazepine treatmentContributions of the GABAA receptor alpha6 subunit to phasic and tonic inhibition revealed by a naturally occurring polymorphism in the alpha6 geneα2-containing GABA(A) receptors: a requirement for midazolam-escalated aggression and social approach in miceA Tribute to Peter H Seeburg (1944-2016): A Founding Father of Molecular Neurobiology.The influence of stress at puberty on mood and learning: role of the α4βδ GABAA receptorBenzodiazepine-induced anxiolysis and reduction of conditioned fear are mediated by distinct GABAA receptor subtypes in miceStudying Cerebellar Circuits by Remote Control of Selected Neuronal Types with GABA(A) ReceptorsNeurosteroid regulation of GABA(A) receptors: Focus on the alpha4 and delta subunits.Hooked on benzodiazepines: GABAA receptor subtypes and addiction.Privileged diazepine compounds and their emergence as bromodomain inhibitors.Cocaine effects on mouse incentive-learning and human addiction are linked to alpha2 subunit-containing GABAA receptors.Low dose acute alcohol effects on GABA A receptor subtypesNovel positive allosteric modulators of GABAA receptors: do subtle differences in activity at alpha1 plus alpha5 versus alpha2 plus alpha3 subunits account for dissimilarities in behavioral effects in rats?A nonequilibrium binary elements-based kinetic model for benzodiazepine regulation of GABAA receptors.Molecular targets and mechanisms for ethanol action in glycine receptorsThe modulatory action of loreclezole at the gamma-aminobutyric acid type A receptor is determined by a single amino acid in the beta 2 and beta 3 subunitInfluence of GABA(A) receptor α subunit isoforms on the benzodiazepine binding siteFlavonoid modulation of GABA(A) receptors.A Multifaceted GABAA Receptor Modulator: Functional Properties and Mechanism of Action of the Sedative-Hypnotic and Recreational Drug Methaqualone (Quaalude)Retrochalcone derivatives are positive allosteric modulators at synaptic and extrasynaptic GABA(A) receptors in vitroGABAA receptors in the posterior, but not anterior, ventral tegmental area mediate Ro15-4513-induced attenuation of binge-like ethanol consumption in C57BL/6J female miceThymol, a constituent of thyme essential oil, is a positive allosteric modulator of human GABA(A) receptors and a homo-oligomeric GABA receptor from Drosophila melanogaster2D IR spectroscopy of histidine: probing side-chain structure and dynamics via backbone amide vibrations.Different residues in the GABAA receptor benzodiazepine binding pocket mediate benzodiazepine efficacy and binding.The role of GABAA receptors in mediating the effects of alcohol in the central nervous system.The dynamic modulation of GABA(A) receptor trafficking and its role in regulating the plasticity of inhibitory synapses.Mechanism of action of benzodiazepines on GABAA receptors.Desformylflustrabromine Modulates α4β2 Neuronal Nicotinic Acetylcholine Receptor High- and Low-Sensitivity Isoforms at Allosteric Clefts Containing the β2 SubunitA new meaning for "Gin & Tonic": tonic inhibition as the target for ethanol action in the brain.Mechanisms of neurosteroid interactions with GABA(A) receptors.
P2860
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P2860
A single histidine in GABAA receptors is essential for benzodiazepine agonist binding
description
1992 թուականի Յունուարին հրատարակուած գիտական յօդուած
@hyw
1992 թվականի հունվարին հրատարակված գիտական հոդված
@hy
article publié dans la revue scientifique Journal of Biological Chemistry
@fr
artículu científicu espublizáu en 1992
@ast
im Januar 1992 veröffentlichter wissenschaftlicher Artikel
@de
scientific journal article
@en
vedecký článok (publikovaný 1992/01/25)
@sk
vědecký článek publikovaný v roce 1992
@cs
wetenschappelijk artikel (gepubliceerd op 1992/01/25)
@nl
наукова стаття, опублікована в січні 1992
@uk
name
A single histidine in GABAA receptors is essential for benzodiazepine agonist binding
@ast
A single histidine in GABAA receptors is essential for benzodiazepine agonist binding
@en
A single histidine in GABAA receptors is essential for benzodiazepine agonist binding
@nl
type
label
A single histidine in GABAA receptors is essential for benzodiazepine agonist binding
@ast
A single histidine in GABAA receptors is essential for benzodiazepine agonist binding
@en
A single histidine in GABAA receptors is essential for benzodiazepine agonist binding
@nl
prefLabel
A single histidine in GABAA receptors is essential for benzodiazepine agonist binding
@ast
A single histidine in GABAA receptors is essential for benzodiazepine agonist binding
@en
A single histidine in GABAA receptors is essential for benzodiazepine agonist binding
@nl
P1476
A single histidine in GABAA receptors is essential for benzodiazepine agonist binding
@en
P2093
H. A. Wieland
H. Lüddens
P304
P407
P577
1992-01-25T00:00:00Z