The malaria parasite's chloroquine resistance transporter is a member of the drug/metabolite transporter superfamily
about
The 'permeome' of the malaria parasite: an overview of the membrane transport proteins of Plasmodium falciparum.Assessment of Plasmodium falciparum resistance to ferroquine (SSR97193) in field isolates and in W2 strain under pressure.Antimalarial drug resistance: An overviewAntimalarial Drug Resistance: Literature Review and Activities and Findings of the ICEMR NetworkThe interplay between drug resistance and fitness in malaria parasitesUDP-galactose and acetyl-CoA transporters as Plasmodium multidrug resistance genesPfCRT and its role in antimalarial drug resistanceGenome-wide compensatory changes accompany drug- selected mutations in the Plasmodium falciparum crt geneIdentification of a mutant PfCRT-mediated chloroquine tolerance phenotype in Plasmodium falciparumOn the mechanism of chloroquine resistance in Plasmodium falciparumFunctional characterization of the Plasmodium falciparum chloroquine-resistance transporter (PfCRT) in transformed Dictyostelium discoideum vesiclesMetabolic QTL analysis links chloroquine resistance in Plasmodium falciparum to impaired hemoglobin catabolismMolecular Mechanisms for Drug Hypersensitivity Induced by the Malaria Parasite's Chloroquine Resistance TransporterInvestigation of the Plasmodium falciparum food vacuole through inducible expression of the chloroquine resistance transporter (PfCRT)Membrane transporters in the relict plastid of malaria parasitesChloroquine transport via the malaria parasite's chloroquine resistance transporterMultiple drugs compete for transport via the Plasmodium falciparum chloroquine resistance transporter at distinct but interdependent sitesChloroquine-resistant isoforms of the Plasmodium falciparum chloroquine resistance transporter acidify lysosomal pH in HEK293 cells more than chloroquine-sensitive isoforms.Characterization of the chloroquine resistance transporter homologue in Toxoplasma gondiiFormation of the food vacuole in Plasmodium falciparum: a potential role for the 19 kDa fragment of merozoite surface protein 1 (MSP1(19))Simplified Reversed Chloroquines To Overcome Malaria Resistance to Quinoline-Based DrugsPlant homologs of the Plasmodium falciparum chloroquine-resistance transporter, PfCRT, are required for glutathione homeostasis and stress responsesQuinine dimers are potent inhibitors of the Plasmodium falciparum chloroquine resistance transporter and are active against quinoline-resistant P. falciparumMutations in pfmdr1 modulate the sensitivity of Plasmodium falciparum to the intrinsic antiplasmodial activity of verapamilReversal agent and linker variants of reversed chloroquines: activities against Plasmodium falciparum.Synthesis, structure-activity relationship, and mode-of-action studies of antimalarial reversed chloroquine compounds.PfCRT and the trans-vacuolar proton electrochemical gradient: regulating the access of chloroquine to ferriprotoporphyrin IX.Transporters involved in resistance to antimalarial drugs.Quantitative genome re-sequencing defines multiple mutations conferring chloroquine resistance in rodent malariaThe toxoplasma apicoplast phosphate translocator links cytosolic and apicoplast metabolism and is essential for parasite survival.1H-NMR metabolite profiles of different strains of Plasmodium falciparum.Lack of association between putative transporter gene polymorphisms in Plasmodium falciparum and chloroquine resistance in imported malaria isolates from AfricaAntimalarial screening via large-scale purification of Plasmodium falciparum Ca2+-ATPase 6 and in vitro studies.Predicting functional and regulatory divergence of a drug resistance transporter gene in the human malaria parasiteAzithromycin plus chloroquine: combination therapy for protection against malaria and sexually transmitted infections in pregnancy.Plasmodium falciparum chloroquine resistance transporter is a H+-coupled polyspecific nutrient and drug exporter.Dictyostelium discoideum expresses a malaria chloroquine resistance mechanism upon transfection with mutant, but not wild-type, Plasmodium falciparum transporter PfCRT.Adaptive evolution of malaria parasites in French Guiana: Reversal of chloroquine resistance by acquisition of a mutation in pfcrtMutations in the Plasmodium falciparum chloroquine resistance transporter, PfCRT, enlarge the parasite's food vacuole and alter drug sensitivities.Malaria drug resistance: new observations and developments.
P2860
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P2860
The malaria parasite's chloroquine resistance transporter is a member of the drug/metabolite transporter superfamily
description
2004 nî lūn-bûn
@nan
2004 թուականի Հոկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2004 թվականի հոտեմբերին հրատարակված գիտական հոդված
@hy
2004年の論文
@ja
2004年論文
@yue
2004年論文
@zh-hant
2004年論文
@zh-hk
2004年論文
@zh-mo
2004年論文
@zh-tw
2004年论文
@wuu
name
The malaria parasite's chloroq ...... bolite transporter superfamily
@ast
The malaria parasite's chloroq ...... bolite transporter superfamily
@en
type
label
The malaria parasite's chloroq ...... bolite transporter superfamily
@ast
The malaria parasite's chloroq ...... bolite transporter superfamily
@en
prefLabel
The malaria parasite's chloroq ...... bolite transporter superfamily
@ast
The malaria parasite's chloroq ...... bolite transporter superfamily
@en
P921
P3181
P356
P1476
The malaria parasite's chloroq ...... bolite transporter superfamily
@en
P304
P3181
P356
10.1093/MOLBEV/MSH205
P407
P577
2004-10-01T00:00:00Z