2-Dialkynyl derivatives of (N)-methanocarba nucleosides: 'Clickable' A(3) adenosine receptor-selective agonists.
about
Polyamidoamine (PAMAM) dendrimer conjugate specifically activates the A3 adenosine receptor to improve post-ischemic/reperfusion function in isolated mouse hearts.Polyamidoamine (PAMAM) dendrimer conjugates of "clickable" agonists of the A3 adenosine receptor and coactivation of the P2Y14 receptor by a tethered nucleotide.GPCR ligand dendrimer (GLiDe) conjugates: adenosine receptor interactions of a series of multivalent xanthine antagonistsAnti-ischemic effects of multivalent dendrimeric A₃ adenosine receptor agonists in cultured cardiomyocytes and in the isolated rat heart.Click modification in the N6 region of A3 adenosine receptor-selective carbocyclic nucleosides for dendrimeric tethering that preserves pharmacophore recognition.Methanocarba ring as a ribose modification in ligands of G protein-coupled purine and pyrimidine receptors: synthetic approaches.Structure-Based Design, Synthesis by Click Chemistry and in Vivo Activity of Highly Selective A3 Adenosine Receptor Agonists.Lighting up G protein-coupled purinergic receptors with engineered fluorescent ligands.Fluorescent ligands for adenosine receptors.Characterization by flow cytometry of fluorescent, selective agonist probes of the A(3) adenosine receptor.Modulation of G protein-coupled adenosine receptors by strategically functionalized agonists and antagonists immobilized on gold nanoparticles.Synthesis of BODIPY derivatives substituted with various bioconjugatable linker groups: a construction kit for fluorescent labeling of receptor ligands.
P2860
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P2860
2-Dialkynyl derivatives of (N)-methanocarba nucleosides: 'Clickable' A(3) adenosine receptor-selective agonists.
description
2009 nî lūn-bûn
@nan
2009 թուականի Դեկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2009 թվականի դեկտեմբերին հրատարակված գիտական հոդված
@hy
2009年の論文
@ja
2009年論文
@yue
2009年論文
@zh-hant
2009年論文
@zh-hk
2009年論文
@zh-mo
2009年論文
@zh-tw
2009年论文
@wuu
name
2-Dialkynyl derivatives of (N) ...... e receptor-selective agonists.
@ast
2-Dialkynyl derivatives of (N) ...... e receptor-selective agonists.
@en
type
label
2-Dialkynyl derivatives of (N) ...... e receptor-selective agonists.
@ast
2-Dialkynyl derivatives of (N) ...... e receptor-selective agonists.
@en
prefLabel
2-Dialkynyl derivatives of (N) ...... e receptor-selective agonists.
@ast
2-Dialkynyl derivatives of (N) ...... e receptor-selective agonists.
@en
P2093
P2860
P1476
2-Dialkynyl derivatives of (N) ...... e receptor-selective agonists.
@en
P2093
Dong Wook Kang
Hans Luecke
Kenneth A Jacobson
Lena S Yoo
Moshe Chinn
Zhan-Guo Gao
P2860
P304
P356
10.1016/J.BMC.2009.12.018
P407
P50
P577
2009-12-11T00:00:00Z