Benzothiadiazides inhibit rapid glutamate receptor desensitization and enhance glutamatergic synaptic currents.
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7-Chloro-3-methyl-3,4-dihydro-2H-1,2,4-benzothiadiazine S,S-dioxide (IDRA 21), a congener of aniracetam, potently abates pharmacologically induced cognitive impairments in patas monkeysCyclothiazide induces seizure behavior in freely moving rats.Cyclothiazide potently inhibits gamma-aminobutyric acid type A receptors in addition to enhancing glutamate responsesTargeting AMPA receptor gating processes with allosteric modulators and mutations7-Chloro-3-methyl-3,4-dihydro-2H-1,2,4-benzothiadiazine S,S-dioxide: a partial modulator of AMPA receptor desensitization devoid of neurotoxicityCyclothiazide induces robust epileptiform activity in rat hippocampal neurons both in vitro and in vivoTuning activation of the AMPA-sensitive GluR2 ion channel by genetic adjustment of agonist-induced conformational changesStability of ligand-binding domain dimer assembly controls kainate receptor desensitizationProbing the Allosteric Modulator Binding Site of GluR2 with Thiazide DerivativesGlutamate receptor ion channels: structure, regulation, and functionMechanisms underlying presynaptic facilitatory effect of cyclothiazide at the calyx of Held of juvenile ratsCyclothiazide-induced persistent increase in respiratory-related activity in vitroShort-term plasticity and auditory processing in the ventral cochlear nucleus of normal and hearing-impaired animalsA low-affinity antagonist reveals saturation and desensitization in mature synapses in the auditory brain stem.Relative roles of different mechanisms of depression at the mouse endbulb of Held.Brominated 7-hydroxycoumarin-4-ylmethyls: photolabile protecting groups with biologically useful cross-sections for two photon photolysisA novel Conus snail polypeptide causes excitotoxicity by blocking desensitization of AMPA receptorsConcentration-jump analysis of voltage-dependent conductances activated by glutamate and kainate in neurons of the avian cochlear nucleus.Calcium regulates vesicle replenishment at the cone ribbon synapse.Effects of cyclothiazide on GluR1/AMPA receptorsStructure and dynamics of AMPA receptor GluA2 in resting, pre-open, and desensitized statesAMPA receptor potentiators: from drug design to cognitive enhancementProconvulsive effect of hydrochlorothiazide in an in vitro rat seizure model.Interaction between positive allosteric modulators and trapping blockers of the NMDA receptor channel.Glutamate regulates intracellular calcium and gene expression in oligodendrocyte progenitors through the activation of DL-alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptors.Inhibitory-excitatory synaptic balance is shifted toward increased excitation in magnocellular neurosecretory cells of heart failure rats.The chemokine growth-related gene product beta protects rat cerebellar granule cells from apoptotic cell death through alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionate receptors.Selective and sustained α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor activation in cerebellum induces dystonia in mice.Allosteric interactions between cyclothiazide and AMPA/kainate receptor antagonists.Screening for AMPA receptor auxiliary subunit specific modulators.Pharmacological treatment with mirtazapine rescues cortical atrophy and respiratory deficits in MeCP2 null mice.Sigma receptors [σRs]: biology in normal and diseased statesA novel class of allosteric modulators of AMPA/Kainate receptors.AMPA receptors promote perivascular glioma invasion via beta1 integrin-dependent adhesion to the extracellular matrix.BDNF-TrkB signaling pathway mediates the induction of epileptiform activity induced by a convulsant drug cyclothiazide.The role of SNP-loop diuretic interactions in hypertension across ethnic groups in HyperGENPAR1 activation induces rapid changes in glutamate uptake and astrocyte morphology.Estimating synaptic parameters from mean, variance, and covariance in trains of synaptic responses.Effects of reduced vesicular filling on synaptic transmission in rat hippocampal neurones.A comparison of release kinetics and glutamate receptor properties in shaping rod-cone differences in EPSC kinetics in the salamander retina.
P2860
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P2860
Benzothiadiazides inhibit rapid glutamate receptor desensitization and enhance glutamatergic synaptic currents.
description
1993 nî lūn-bûn
@nan
1993 թուականի Սեպտեմբերին հրատարակուած գիտական յօդուած
@hyw
1993 թվականի սեպտեմբերին հրատարակված գիտական հոդված
@hy
1993年の論文
@ja
1993年論文
@yue
1993年論文
@zh-hant
1993年論文
@zh-hk
1993年論文
@zh-mo
1993年論文
@zh-tw
1993年论文
@wuu
name
Benzothiadiazides inhibit rapi ...... utamatergic synaptic currents.
@ast
Benzothiadiazides inhibit rapi ...... utamatergic synaptic currents.
@en
Benzothiadiazides inhibit rapi ...... utamatergic synaptic currents.
@nl
type
label
Benzothiadiazides inhibit rapi ...... utamatergic synaptic currents.
@ast
Benzothiadiazides inhibit rapi ...... utamatergic synaptic currents.
@en
Benzothiadiazides inhibit rapi ...... utamatergic synaptic currents.
@nl
prefLabel
Benzothiadiazides inhibit rapi ...... utamatergic synaptic currents.
@ast
Benzothiadiazides inhibit rapi ...... utamatergic synaptic currents.
@en
Benzothiadiazides inhibit rapi ...... utamatergic synaptic currents.
@nl
P1476
Benzothiadiazides inhibit rapi ...... lutamatergic synaptic currents
@en
P2093
P304
P356
10.1523/JNEUROSCI.13-09-03904.1993
P407
P577
1993-09-01T00:00:00Z