High-throughput screening approaches for investigating drug metabolism and pharmacokinetics.
about
Lead Optimization in Discovery Drug Metabolism and Pharmacokinetics/Case study: The Hepatitis C Virus (HCV) Protease Inhibitor SCH 503034Toxicity testing in the 21st century: a vision and a strategyHigh-throughput 1,536-well fluorescence polarization assays for α(1)-acid glycoprotein and human serum albumin bindingAn ultra high-throughput, whole-animal screen for small molecule modulators of a specific genetic pathway in Caenorhabditis elegansEltrombopag: the discovery of a second generation thrombopoietin-receptor agonist.Strategies to improve oral drug bioavailability.Phenylalanine 4-monooxygenase and the role of endobiotic metabolism enzymes in xenobiotic biotransformation.Prediction of human pharmacokinetics--evaluation of methods for prediction of hepatic metabolic clearance.Rapid in vivo oral screening in rats: reliability, acceptance criteria, and filtering efficiency.Progress toward virtual screening for drug side effects.Characterization of mixtures of recombinant human cytochrome p450s as a screening model for metabolic stability in drug discovery.In silico insights: chemical and structural characteristics associated with uridine diphosphate-glucuronosyltransferase substrate selectivity.
P2860
Q27489828-88CEC354-4E0F-447C-9067-C9B9346C1AA1Q27921848-5A51CE3F-FACD-461A-9484-62BB40792C90Q28483928-4EF572EA-1AA5-4281-85E1-2F73EE731E6FQ28487176-7FB243A5-B6E9-43B0-A018-5ABD8A969523Q33406379-75D09134-5A69-4945-8A50-C67896E1F720Q36316751-CC202EEF-2CEE-4C6B-96E3-753D8C949B8CQ37571937-38C25E7A-946B-4433-8841-B4EA092309A6Q39805145-E64AAF07-60EC-4986-909A-760561EFBFA4Q41960216-0F47554C-4A7A-43A0-9DB7-11A68C37BCD5Q44125156-46D0A0E4-DC0A-4240-9415-1BA0BE605EF6Q44191382-71316E94-CAFE-4264-9C69-EF8CA8381606Q44695257-C7A6B52F-64DC-4C97-8689-0A3DB67434BE
P2860
High-throughput screening approaches for investigating drug metabolism and pharmacokinetics.
description
2001 nî lūn-bûn
@nan
2001 թուականի Օգոստոսին հրատարակուած գիտական յօդուած
@hyw
2001 թվականի օգոստոսին հրատարակված գիտական հոդված
@hy
2001年の論文
@ja
2001年論文
@yue
2001年論文
@zh-hant
2001年論文
@zh-hk
2001年論文
@zh-mo
2001年論文
@zh-tw
2001年论文
@wuu
name
High-throughput screening appr ...... tabolism and pharmacokinetics.
@ast
High-throughput screening appr ...... tabolism and pharmacokinetics.
@en
High-throughput screening appr ...... tabolism and pharmacokinetics.
@nl
type
label
High-throughput screening appr ...... tabolism and pharmacokinetics.
@ast
High-throughput screening appr ...... tabolism and pharmacokinetics.
@en
High-throughput screening appr ...... tabolism and pharmacokinetics.
@nl
prefLabel
High-throughput screening appr ...... tabolism and pharmacokinetics.
@ast
High-throughput screening appr ...... tabolism and pharmacokinetics.
@en
High-throughput screening appr ...... tabolism and pharmacokinetics.
@nl
P2860
P1433
P1476
High-throughput screening appr ...... tabolism and pharmacokinetics.
@en
P2093
S A Roberts
P2860
P304
P356
10.1080/00498250110060978
P407
P577
2001-08-01T00:00:00Z