Aiming for allosterism: Evaluation of allosteric modulators of CB1 in a neuronal model.
about
Allosteric Modulation: An Alternate Approach Targeting the Cannabinoid CB1 Receptor.In silico mapping of allosteric ligand binding sites in type-1 cannabinoid receptor.The great divide: Separation between in vitro and in vivo effects of PSNCBAM-based CB1 receptor allosteric modulators.Preclinical Studies of Cannabinoid Reward, Treatments for Cannabis Use Disorder, and Addiction-Related Effects of Cannabinoid Exposure.Positive Allosteric Modulation of Cannabinoid Receptor Type 1 Suppresses Pathological Pain Without Producing Tolerance or Dependence.Leveraging allostery to improve G protein-coupled receptor (GPCR)-directed therapeutics: cannabinoid receptor 1 as discovery target.TRP channels as novel targets for endogenous ligands: focus on endocannabinoids and nociceptive signalling.Modulation of CB1 cannabinoid receptor by allosteric ligands: Pharmacology and therapeutic opportunities.Pepcan-12 (RVD-hemopressin) is a CB2 receptor positive allosteric modulator constitutively secreted by adrenals and in liver upon tissue damage.Allosteric Modulators of the CB1 Cannabinoid Receptor: A Structural Update Review.Assessing Allosteric Modulation of CB1 at the Receptor and Cellular Levels.Enantiomer-specific positive allosteric modulation of CB1 signaling in autaptic hippocampal neurons.The endocannabinoid system in guarding against fear, anxiety and stress.Cannabidiol attenuates seizures and social deficits in a mouse model of Dravet syndrome.
P2860
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P2860
Aiming for allosterism: Evaluation of allosteric modulators of CB1 in a neuronal model.
description
2015 nî lūn-bûn
@nan
2015年の論文
@ja
2015年論文
@yue
2015年論文
@zh-hant
2015年論文
@zh-hk
2015年論文
@zh-mo
2015年論文
@zh-tw
2015年论文
@wuu
2015年论文
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2015年论文
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name
Aiming for allosterism: Evaluation of allosteric modulators of CB1 in a neuronal model.
@ast
Aiming for allosterism: Evaluation of allosteric modulators of CB1 in a neuronal model.
@en
type
label
Aiming for allosterism: Evaluation of allosteric modulators of CB1 in a neuronal model.
@ast
Aiming for allosterism: Evaluation of allosteric modulators of CB1 in a neuronal model.
@en
prefLabel
Aiming for allosterism: Evaluation of allosteric modulators of CB1 in a neuronal model.
@ast
Aiming for allosterism: Evaluation of allosteric modulators of CB1 in a neuronal model.
@en
P2093
P2860
P1476
Aiming for allosterism: Evaluation of allosteric modulators of CB1 in a neuronal model
@en
P2093
Alex Straiker
Anne Gibson
Danielle Yin
José Mitjavila
P2860
P304
P356
10.1016/J.PHRS.2015.07.017
P50
P577
2015-07-23T00:00:00Z