Phospho-MurNAc-pentapeptide translocase (MraY) as a target for antibacterial agents and antibacterial proteins.
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The Membrane Steps of Bacterial Cell Wall Synthesis as Antibiotic TargetsCore Steps of Membrane-Bound Peptidoglycan Biosynthesis: Recent Advances, Insight and OpportunitiesCrystal structure of a peptidoglycan glycosyltransferase suggests a model for processive glycan chain synthesisCrystal Structure of MraY, an Essential Membrane Enzyme for Bacterial Cell Wall SynthesisSpecificity Determinants for Lysine Incorporation in Staphylococcus aureus Peptidoglycan as Revealed by the Structure of a MurE Enzyme Ternary ComplexPreparative scale cell-free production and quality optimization of MraY homologues in different expression modesStructural insights into inhibition of lipid I production in bacterial cell wall synthesis.Treatment of Clostridium difficile infection using SQ641, a capuramycin analogue, increases post-treatment survival and improves clinical measures of disease in a murine model.Inhibition of Escherichia coli glycosyltransferase MurG and Mycobacterium tuberculosis Gal transferase by uridine-linked transition state mimics.Amino acid motifs in natural products: synthesis of O-acylated derivatives of (2S,3S)-3-hydroxyleucine.Analysis of a dual domain phosphoglycosyl transferase reveals a ping-pong mechanism with a covalent enzyme intermediate.A high-throughput screen for directed evolution of the natural product sulfotransferase LipB.Biosynthesis of a water-soluble lipid I analogue and a convenient assay for translocase I.Synthesis of ureidomuraymycidine derivatives for structure-activity relationship studies of muraymycins.A reliable Pd-mediated hydrogenolytic deprotection of BOM group of uridine ureido nitrogenA new protecting group and linker for uridine ureido nitrogen.Fluorescence-based assay for polyprenyl phosphate-GlcNAc-1-phosphate transferase (WecA) and identification of novel antimycobacterial WecA inhibitors.Novel approaches to developing new antibiotics for bacterial infections.Lipid Requirements for the Enzymatic Activity of MraY Translocases and in Vitro Reconstitution of the Lipid II Synthesis PathwayThe biosynthesis of peptidoglycan lipid-linked intermediates.Effectiveness of F18+ Fimbrial Antigens Released by a Novel Autolyzed Salmonella Expression System as a Vaccine Candidate against Lethal F18+ STEC Infection.Therapeutic efficacy of SQ641-NE against Mycobacterium tuberculosis.Improved synthesis of capuramycin and its analogues.Challenges and opportunities in developing novel drugs for TB.Update on carbohydrate-containing antibacterial agents.Concise synthesis of capuramycin.Synthesis and Biological Evaluation of Muraymycin Analogues Active against Anti-Drug-Resistant Bacteria.Chemical modification of capuramycins to enhance antibacterial activityExpansion of Antibacterial Spectrum of Muraymycins toward Pseudomonas aeruginosa.N-Acetylglucosamine-1-phosphate transferase, WecA, as a validated drug target in Mycobacterium tuberculosis.Functional and kinetic analysis of the phosphotransferase CapP conferring selective self-resistance to capuramycin antibiotics.Ligand Shaping in Induced Fit Docking of MraY Inhibitors. Polynomial Discriminant and Laplacian Operator as Biological Activity Descriptors.Effect of uridine protecting groups on the diastereoselectivity of uridine-derived aldehyde 5'-alkynylation.Structural Investigation of Park's Nucleotide on Bacterial Translocase MraY: Discovery of Unexpected MraY Inhibitors.Genetic analysis of MraY inhibition by the phiX174 protein EMinimal requirements for inhibition of MraY by lysis protein E from bacteriophage ΦX174.In vitro antimicrobial activities of capuramycin analogues against non-tuberculous mycobacteriaUndecaprenyl phosphate metabolism in Gram-negative and Gram-positive bacteria.Insights into the Target Interaction of Naturally Occurring Muraymycin Nucleoside Antibiotics.A Three-Ring Circus: Metabolism of the Three Proteogenic Aromatic Amino Acids and Their Role in the Health of Plants and Animals.
P2860
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P2860
Phospho-MurNAc-pentapeptide translocase (MraY) as a target for antibacterial agents and antibacterial proteins.
description
2006 nî lūn-bûn
@nan
2006年の論文
@ja
2006年論文
@yue
2006年論文
@zh-hant
2006年論文
@zh-hk
2006年論文
@zh-mo
2006年論文
@zh-tw
2006年论文
@wuu
2006年论文
@zh
2006年论文
@zh-cn
name
Phospho-MurNAc-pentapeptide tr ...... ts and antibacterial proteins.
@ast
Phospho-MurNAc-pentapeptide tr ...... ts and antibacterial proteins.
@en
type
label
Phospho-MurNAc-pentapeptide tr ...... ts and antibacterial proteins.
@ast
Phospho-MurNAc-pentapeptide tr ...... ts and antibacterial proteins.
@en
prefLabel
Phospho-MurNAc-pentapeptide tr ...... ts and antibacterial proteins.
@ast
Phospho-MurNAc-pentapeptide tr ...... ts and antibacterial proteins.
@en
P1476
Phospho-MurNAc-pentapeptide tr ...... ts and antibacterial proteins.
@en
P2093
Adrian J Lloyd
Timothy D H Bugg
P304
P356
10.2174/187152606784112128
P577
2006-06-01T00:00:00Z