The macrocyclic tetrapeptide [D-Trp]CJ-15,208 produces short-acting κ opioid receptor antagonism in the CNS after oral administration.

The macrocyclic tetrapeptide [D-Trp]CJ-15,208 produces short-acting κ opioid receptor antagonism in the CNS after oral administration.

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http://www.wikidata.org/entity/Q36836438
Role of kappa-opioid receptors in stress and anxiety-related behavior.Characterization of BU09059: a novel potent selective κ-receptor antagonistStress-Induced Reinstatement of Drug Seeking: 20 Years of Progress.Alanine analogues of [D-Trp]CJ-15,208: novel opioid activity profiles and prevention of drug- and stress-induced reinstatement of cocaine-seeking behaviour.Selective κ receptor partial agonist HS666 produces potent antinociception without inducing aversion after i.c.v. administration in mice.Didehydro-cortistatin A inhibits HIV-1 Tat mediated neuroinflammation and prevents potentiation of cocaine reward in Tat transgenic miceDirect Phenotypic Screening in Mice: Identification of Individual, Novel Antinociceptive Compounds from a Library of 734,821 Pyrrolidine Bis-piperazines.Synthesis and characterization of a dual kappa-delta opioid receptor agonist analgesic blocking cocaine reward behaviorCombined administration of buprenorphine and naltrexone produces antidepressant-like effects in miceDevelopment of a robust, sensitive and selective liquid chromatography-tandem mass spectrometry assay for the quantification of the novel macrocyclic peptide kappa opioid receptor antagonist [D-Trp]CJ-15,208 in plasma and application to an initial pA role for kappa-, but not mu-opioid, receptor activation in acute food deprivation-induced reinstatement of heroin seeking in rats.Tryptophan-Containing Non-Cationizable Opioid Peptides - a new chemotype with unusual structure and in vivo activity.Macrocyclic peptides decrease c-Myc protein levels and reduce prostate cancer cell growth.
P2860

The macrocyclic tetrapeptide [D-Trp]CJ-15,208 produces short-acting κ opioid receptor antagonism in the CNS after oral administration.

Item
http://www.wikidata.org/entity/Q36836438
description
2013 nî lūn-bûn
@nan
2013年の論文
@ja
2013年論文
@yue
2013年論文
@zh-hant
2013年論文
@zh-hk
2013年論文
@zh-mo
2013年論文
@zh-tw
2013年论文
@wuu
2013年论文
@zh
2013年论文
@zh-cn
name
The macrocyclic tetrapeptide [ ...... CNS after oral administration.
@en
type
label
The macrocyclic tetrapeptide [ ...... CNS after oral administration.
@en
prefLabel
The macrocyclic tetrapeptide [ ...... CNS after oral administration.
@en
P1433
P1476
P2093
P2860
P304
P31
P356
P407
P433
P478
P577
P698
P932
P356
P1433
P1476
The macrocyclic tetrapeptide [ ...... CNS after oral administration.
@en
P2093
P2860
P304
P31
P356
P407
P433
P478
P577
P698
P932