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Phytochemicals and Biogenic Metallic Nanoparticles as Anticancer AgentsStabilizing versus destabilizing the microtubules: a double-edge sword for an effective cancer treatment option?Structural Insights into the Pharmacophore of Vinca Domain Inhibitors of MicrotubulesEGF-induced centrosome separation promotes mitotic progression and cell survival.The pathobiology of glioma tumorsSynthesis, antimitotic and antivascular activity of 1-(3',4',5'-trimethoxybenzoyl)-3-arylamino-5-amino-1,2,4-triazoles.Design, synthesis and biological evaluation of 3,5-disubstituted 2-amino thiophene derivatives as a novel class of antitumor agents.Microtubular stability affects pVHL-mediated regulation of HIF-1alpha via the p38/MAPK pathway in hypoxic cardiomyocytes.Synthesis and discovery of water-soluble microtubule targeting agents that bind to the colchicine site on tubulin and circumvent Pgp mediated resistanceMathematical modeling of microtubule dynamics: insights into physiology and disease.Middle infrared radiation induces G2/M cell cycle arrest in A549 lung cancer cellsSuperior antitumor activity of nanoparticle albumin-bound paclitaxel in experimental gastric cancer.Convergent synthesis and biological evaluation of 2-amino-4-(3',4',5'-trimethoxyphenyl)-5-aryl thiazoles as microtubule targeting agents.Drugs that target dynamic microtubules: a new molecular perspectiveRole of Drp1, a key mitochondrial fission protein, in neuropathic pain.Role of Ran-regulated nuclear-cytoplasmic trafficking of pVHL in the regulation of microtubular stability-mediated HIF-1α in hypoxic cardiomyocytesUtility of vascular endothelial growth factor inhibitors in the treatment of ovarian cancer: from concept to application.Synthesis and antitumor molecular mechanism of agents based on amino 2-(3',4',5'-trimethoxybenzoyl)benzo[b]furan: inhibition of tubulin and induction of apoptosis.Design and synthesis of imidazo[2,1-b]thiazole-chalcone conjugates: microtubule-destabilizing agents.Development of a novel class of tubulin inhibitor from desmosdumotin B with a hydroxylated bicyclic B-ringBreast cancer medications and vision: effects of treatments for early-stage disease.One-pot synthesis and biological evaluation of 2-pyrrolidinyl-4-amino-5-(3',4',5'-trimethoxybenzoyl)thiazole: a unique, highly active antimicrotubule agent.Synthesis and evaluation of 1,5-disubstituted tetrazoles as rigid analogues of combretastatin A-4 with potent antiproliferative and antitumor activity.The synergic effect of vincristine and vorinostat in leukemia in vitro and in vivo.Evaluation of activity and combination strategies with the microtubule-targeting drug sagopilone in breast cancer cell lines.Discovery and optimization of a series of 2-aryl-4-amino-5-(3',4',5'-trimethoxybenzoyl)thiazoles as novel anticancer agents.A phase I trial of MK-0731, a kinesin spindle protein (KSP) inhibitor, in patients with solid tumors.Medicinal Plants: Their Use in Anticancer Treatment.Synthesis and biological evaluation of 2-substituted-4-(3',4',5'-trimethoxyphenyl)-5-aryl thiazoles as anticancer agents.Overview of major classes of plant-derived anticancer drugsFrom fighting depression to conquering tumors: a novel tricyclic thiazepine compound as a tubulin polymerization inhibitorThe microtubule stabilizer patupilone counteracts ionizing radiation-induced matrix metalloproteinase activity and tumor cell invasionRegulatory polymorphisms in β-tubulin IIa are associated with paclitaxel-induced peripheral neuropathy.Predicting cancer-relevant proteins using an improved molecular similarity ensemble approach.Structure-activity relationship and in vitro and in vivo evaluation of the potent cytotoxic anti-microtubule agent N-(4-methoxyphenyl)-N,2,6-trimethyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-aminium chloride and its analogues as antitumor agents.In vitro and in vivo anti-tumour effects of MPT0B014, a novel derivative aroylquinoline, and in combination with erlotinib in human non-small-cell lung cancer cells.Parthenolide and costunolide reduce microtentacles and tumor cell attachment by selectively targeting detyrosinated tubulin independent from NF-κB inhibition.Curcumin targets breast cancer stem-like cells with microtentacles that persist in mammospheres and promote reattachment.The medicinal potential of promising marine macrolides with anticancer activity.The tubulin colchicine domain: a molecular modeling perspective.
P2860
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P2860
description
article científic
@ca
article scientifique
@fr
articolo scientifico
@it
artigo científico
@pt
bilimsel makale
@tr
scientific article published on 30 December 2008
@en
vedecký článok
@sk
vetenskaplig artikel
@sv
videnskabelig artikel
@da
vědecký článek
@cs
name
Microtubule dynamics as a target in oncology.
@en
Microtubule dynamics as a target in oncology.
@nl
type
label
Microtubule dynamics as a target in oncology.
@en
Microtubule dynamics as a target in oncology.
@nl
prefLabel
Microtubule dynamics as a target in oncology.
@en
Microtubule dynamics as a target in oncology.
@nl
P2093
P2860
P1476
Microtubule dynamics as a target in oncology.
@en
P2093
April L Risinger
Francis J Giles
Susan L Mooberry
P2860
P304
P356
10.1016/J.CTRV.2008.11.001
P577
2008-12-30T00:00:00Z