Identification of novel, exosite-binding matrix metalloproteinase-13 inhibitor scaffolds.
about
Simple Pseudo-dipeptides with a P2' Glutamate: A NOVEL INHIBITOR FAMILY OF MATRIX METALLOPROTEASES AND OTHER METZINCINSSAR Studies of Exosite-Binding Substrate-Selective Inhibitors of A Disintegrin And Metalloprotease 17 (ADAM17) and Application as Selective in Vitro Probes.Discovery of novel inhibitors of a disintegrin and metalloprotease 17 (ADAM17) using glycosylated and non-glycosylated substrates.Characterization of selective exosite-binding inhibitors of matrix metalloproteinase 13 that prevent articular cartilage degradation in vitro.New strategies for targeting matrix metalloproteinasesThe history of matrix metalloproteinases: milestones, myths, and misperceptions.Potential clinical implications of recent matrix metalloproteinase inhibitor design strategiesActivity of ADAM17 (a disintegrin and metalloprotease 17) is regulated by its noncatalytic domains and secondary structure of its substrates.Matrix metalloproteinase inhibitors: a patent review (2011 - 2013).Clinical implications of compounds designed to inhibit ECM-modifying metalloproteinases.Recent Research Advances in Selective Matrix Metalloproteinase-13 Inhibitors as Anti-Osteoarthritis Agents.Molecular Recognition of the Catalytic Zinc(II) Ion in MMP-13: Structure-Based Evolution of an Allosteric Inhibitor to Dual Binding Mode Inhibitors with Improved Lipophilic Ligand Efficiencies.Strategic targeting of multiple water-mediated interactions: a concise and rational structure-based design approach to potent and selective MMP-13 inhibitorsThe synthesis and application of Fmoc-Lys(5-Fam) building blocks.
P2860
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P2860
Identification of novel, exosite-binding matrix metalloproteinase-13 inhibitor scaffolds.
description
2011 nî lūn-bûn
@nan
2011年の論文
@ja
2011年論文
@yue
2011年論文
@zh-hant
2011年論文
@zh-hk
2011年論文
@zh-mo
2011年論文
@zh-tw
2011年论文
@wuu
2011年论文
@zh
2011年论文
@zh-cn
name
Identification of novel, exosite-binding matrix metalloproteinase-13 inhibitor scaffolds.
@en
type
label
Identification of novel, exosite-binding matrix metalloproteinase-13 inhibitor scaffolds.
@en
prefLabel
Identification of novel, exosite-binding matrix metalloproteinase-13 inhibitor scaffolds.
@en
P2093
P2860
P1476
Identification of novel, exosite-binding matrix metalloproteinase-13 inhibitor scaffolds
@en
P2093
Etzer Darout
Gregg B Fields
Janelle Lauer
Joshua Roth
Peter Hodder
William R Roush
P2860
P304
P356
10.1016/J.BMCL.2011.09.077
P407
P577
2011-09-22T00:00:00Z