Taste, a new incentive to switch to (R)-praziquantel in schistosomiasis treatment
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Open science is a research acceleratorResolution of praziquantelSingle Versus Double Dose Praziquantel Comparison on Efficacy and Schistosoma mansoni Re-Infection in Preschool-Age Children in Uganda: A Randomized Controlled TrialPharmacokinetic Study of Praziquantel Enantiomers and Its Main Metabolite R-trans-4-OH-PZQ in Plasma, Blood and Dried Blood Spots in Opisthorchis viverrini-Infected PatientsStructure-Bioactivity Relationship for Benzimidazole Thiophene Inhibitors of Polo-Like Kinase 1 (PLK1), a Potential Drug Target in Schistosoma mansoniOpen source drug discovery - a limited tutorialPutting the treatment of paediatric schistosomiasis into context.Treatment of intestinal schistosomiasis in Ugandan preschool children: best diagnosis, treatment efficacy and side-effects, and an extended praziquantel dosing poleDesign and synthesis of molecular probes for the determination of the target of the anthelmintic drug praziquantel.Closing the praziquantel treatment gap: new steps in epidemiological monitoring and control of schistosomiasis in African infants and preschool-aged children.Activity of praziquantel enantiomers and main metabolites against Schistosoma mansoni.Metabolic profiling of praziquantel enantiomers.Praziquantel in a clay nanoformulation shows more bioavailability and higher efficacy against murine Schistosoma mansoni infection.The cytotoxicity study of praziquantel enantiomersTHE SUSCEPTIBILITY OF RECENT ISOLATES OF Schistosoma mansoni TO PRAZIQUANTEL.Praziquantel: its use in control of schistosomiasis in sub-Saharan Africa and current research needs.Antiparasitic drugs for paediatrics: systematic review, formulations, pharmacokinetics, safety, efficacy and implications for control.Diagnosis and treatment of schistosomiasis in children in the era of intensified control.In vitro and in vivo activity of R- and S- praziquantel enantiomers and the main human metabolite trans-4-hydroxy-praziquantel against Schistosoma haematobium.What is the mechanism of action of praziquantel and how might resistance strike?Praziquantel for Schistosomiasis: Single-Drug Metabolism Revisited, Mode of Action, and Resistance.Phenotypic, chemical and functional characterization of cyclic nucleotide phosphodiesterase 4 (PDE4) as a potential anthelmintic drug target.Enhancing the usefulness of cross dehydrogenative coupling reactions with a removable protecting group.Synthesis and SAR studies of praziquantel derivatives with activity against Schistosoma japonicum.The anthelmintic praziquantel is a human serotoninergic G-protein-coupled receptor ligand.Validated capillary electrophoretic method for the enantiomeric quality control of R-praziquantel.Accelerating the semisynthesis of alkaloid-based drugs through metabolic engineering.Drug Repurposing for Schistosomiasis: Combinations of Drugs or Biomolecules.Activation of host transient receptor potential (TRP) channels by praziquantel stereoisomers.A Rapid Appraisal of Factors Influencing Praziquantel Treatment Compliance in Two Communities Endemic for Schistosomiasis in Côte d'IvoireExtrapolation of praziquantel pharmacokinetics to a pediatric population: a cautionary taleA comparison of the palatability of racemic praziquantel and its two enantioseparated isomers in yellowtail kingfish Seriola lalandi (Valenciennes, 1833)
P2860
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P2860
Taste, a new incentive to switch to (R)-praziquantel in schistosomiasis treatment
description
2009 nî lūn-bûn
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2009 թուականին հրատարակուած գիտական յօդուած
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2009 թվականին հրատարակված գիտական հոդված
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2009年の論文
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2009年論文
@yue
2009年論文
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2009年論文
@zh-hk
2009年論文
@zh-mo
2009年論文
@zh-tw
2009年论文
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name
Taste, a new incentive to switch to (R)-praziquantel in schistosomiasis treatment
@ast
Taste, a new incentive to switch to (R)-praziquantel in schistosomiasis treatment
@en
Taste, a new incentive to switch to (R)-praziquantel in schistosomiasis treatment
@en-gb
Taste, a new incentive to switch to (R)-praziquantel in schistosomiasis treatment
@nl
type
label
Taste, a new incentive to switch to (R)-praziquantel in schistosomiasis treatment
@ast
Taste, a new incentive to switch to (R)-praziquantel in schistosomiasis treatment
@en
Taste, a new incentive to switch to (R)-praziquantel in schistosomiasis treatment
@en-gb
Taste, a new incentive to switch to (R)-praziquantel in schistosomiasis treatment
@nl
prefLabel
Taste, a new incentive to switch to (R)-praziquantel in schistosomiasis treatment
@ast
Taste, a new incentive to switch to (R)-praziquantel in schistosomiasis treatment
@en
Taste, a new incentive to switch to (R)-praziquantel in schistosomiasis treatment
@en-gb
Taste, a new incentive to switch to (R)-praziquantel in schistosomiasis treatment
@nl
P2093
P2860
P3181
P1476
Taste, a new incentive to switch to (R)-praziquantel in schistosomiasis treatment
@en
P2093
Christian Miculka
Dieter Schollmeyer
Harald Sekljic
Heiko Bothe
Stefan Fuchs
Thorsten Meyer
P2860
P3181
P356
10.1371/JOURNAL.PNTD.0000357
P407
P577
2009-01-01T00:00:00Z