X-ray crystallography: Assessment and validation of protein-small molecule complexes for drug discovery.
about
Charting a Path to Success in Virtual ScreeningX-ray crystallography over the past decade for novel drug discovery - where are we heading next?The future of crystallography in drug discovery.Databases, Repositories, and Other Data Resources in Structural Biology.A public database of macromolecular diffraction experiments.Fitmunk: improving protein structures by accurate, automatic modeling of side-chain conformations.Magnesium-binding architectures in RNA crystal structures: validation, binding preferences, classification and motif detection.Data to knowledge: how to get meaning from your result.Validation of metal-binding sites in macromolecular structures with the CheckMyMetal web server.Protein crystallography for aspiring crystallographers or how to avoid pitfalls and traps in macromolecular structure determination.Metformin impairs glucose consumption and survival in Calu-1 cells by direct inhibition of hexokinase-II.Accurate macromolecular crystallographic refinement: incorporation of the linear scaling, semiempirical quantum-mechanics program DivCon into the PHENIX refinement packageMg2+ ions: do they bind to nucleobase nitrogens?Mapping a protein recognition centre with chiral photoactive ligands. An integrated approach combining photophysics, reactivity, proteomics and molecular dynamics simulation studiesLatest developments in molecular docking: 2010-2011 in review.Molstack - interactive visualization tool for presentation, interpretation, and validation of macromolecules and electron density maps.Conformational energy range of ligands in protein crystal structures: The difficult quest for accurate understanding.Ligand fitting with CCP4.Automated identification of crystallographic ligands using sparse-density representations.Handling ligands with Coot.Chroman-4-One Derivatives Targeting Pteridine Reductase 1 and Showing Anti-Parasitic Activity.Assigning crystallographic electron densities with free energy calculations-The case of the fluoride channel Fluc.Influence of Na+ and Mg2+ ions on RNA structures studied with molecular dynamics simulations.
P2860
Q26779035-E20A451C-236B-40CD-85EB-59F6290A53FAQ26801307-FD1907BE-4719-49F5-AD8E-A5461802A9F9Q28655467-2AE97BB7-7993-413D-8718-26615761339EQ30252226-B0A226A1-CA84-4E58-BCC5-1569A961F7F3Q30275421-A4525454-CB6C-4442-8177-909FF4D03B7AQ30277311-F83A5522-A06D-4F2F-946A-13AEB60B4266Q30300321-BD94C590-D7C5-4F52-B9D6-54A5869ABFE3Q30300912-3C81CDED-C751-4F68-853A-C4C48B437BF3Q30357072-1092F8C5-32C0-4958-8337-486D75084D19Q30409760-9FE08907-AF57-4633-80B4-E6C16DC904F6Q30540902-DA6022AC-D234-42DD-8B17-921FE94DBCA2Q30577677-D21FA878-8ECC-40AE-9883-8F5922FEE8A4Q31147206-06287CD5-6288-4943-A99F-098C672FA6ECQ36383970-E83675DF-B997-4F32-B6D3-9C4A5A18F92BQ38092807-BF64BEB1-8AC5-4D83-BAE6-646AFCE8F68DQ38620864-8AC5D952-EEE3-4AD8-94F4-DD2F21DEBEE8Q38944603-C45C1293-812C-4F28-8864-D799931CC0A1Q41900627-BE8CEAD9-A00D-46D4-A491-1A929D8645F1Q42111041-42D1845F-A2B1-4679-80BE-0640D2FCD65EQ42552372-BD735227-D5C1-4BCC-8AB6-6D0D507493F0Q51102354-111F85E8-CEFB-442C-BAA7-7844C6520D77Q55092949-799F46CF-303C-4145-91D3-13F52A071F79Q55253163-5559E4A3-A384-4873-9810-CC7D68D1E4AB
P2860
X-ray crystallography: Assessment and validation of protein-small molecule complexes for drug discovery.
description
2011 nî lūn-bûn
@nan
2011 թուականի Օգոստոսին հրատարակուած գիտական յօդուած
@hyw
2011 թվականի օգոստոսին հրատարակված գիտական հոդված
@hy
2011年の論文
@ja
2011年論文
@yue
2011年論文
@zh-hant
2011年論文
@zh-hk
2011年論文
@zh-mo
2011年論文
@zh-tw
2011年论文
@wuu
name
X-ray crystallography: Assessm ...... complexes for drug discovery.
@ast
X-ray crystallography: Assessm ...... complexes for drug discovery.
@en
X-ray crystallography: assessm ...... e complexes for drug discovery
@nl
type
label
X-ray crystallography: Assessm ...... complexes for drug discovery.
@ast
X-ray crystallography: Assessm ...... complexes for drug discovery.
@en
X-ray crystallography: assessm ...... e complexes for drug discovery
@nl
prefLabel
X-ray crystallography: Assessm ...... complexes for drug discovery.
@ast
X-ray crystallography: Assessm ...... complexes for drug discovery.
@en
X-ray crystallography: assessm ...... e complexes for drug discovery
@nl
P2860
P50
P1476
X-ray crystallography: Assessm ...... complexes for drug discovery.
@en
P2093
David R Cooper
P2860
P304
P356
10.1517/17460441.2011.585154
P407
P577
2011-08-01T00:00:00Z