The Effects of CapZ Peptide (TRTK-12) Binding to S100B–Ca2+ as Examined by NMR and X-ray Crystallography
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In vitro screening and structural characterization of inhibitors of the S100B-p53 interactionStructure of a C-terminal AHNAK peptide in a 1:2:2 complex with S100A10 and an acetylated N-terminal peptide of annexin A2Asymmetric Mode of Ca2+-S100A4 Interaction with Nonmuscle Myosin IIA Generates Nanomolar Affinity Required for Filament RemodelingAn Interplay of S-Nitrosylation and Metal Ion Binding for Astrocytic S100B ProteinThe relation of the X-ray B-factor to protein dynamics: insights from recent dynamic solid-state NMR data.The design and delivery of a thermally responsive peptide to inhibit S100B-mediated neurodegenerationComplex formation between S100B protein and the p90 ribosomal S6 kinase (RSK) in malignant melanoma is calcium-dependent and inhibits extracellular signal-regulated kinase (ERK)-mediated phosphorylation of RSKModulation of quaternary structure of S100 proteins by calcium ions.Covalent small molecule inhibitors of Ca(2+)-bound S100B.Binding of two intrinsically disordered peptides to a multi-specific protein: a combined Monte Carlo and molecular dynamics studyGlial S100B protein modulates mutant ataxin-1 aggregation and toxicity: TRTK12 peptide, a potential candidate for SCA1 therapyStructural insights into the binding of the human receptor for advanced glycation end products (RAGE) by S100B, as revealed by an S100B-RAGE-derived peptide complex.Small Molecule Inhibitors of Ca(2+)-S100B Reveal Two Protein Conformations.Target binding to S100B reduces dynamic properties and increases Ca(2+)-binding affinity for wild type and EF-hand mutant proteins.Functions of S100 proteins.Novel protein-inhibitor interactions in site 3 of Ca(2+)-bound S100B as discovered by X-ray crystallography.Penetrating the cell membrane, thermal targeting and novel anticancer drugs: the development of thermally targeted, elastin-like polypeptide cancer therapeutics.Identification of calcium-independent and calcium-enhanced binding between S100B and the dopamine D2 receptorThe S100A10-annexin A2 complex provides a novel asymmetric platform for membrane repair.Structural and thermodynamic characterization of the recognition of the S100-binding peptides TRTK12 and p53 by calmodulinThermodynamic and kinetic analysis of peptides derived from CapZ, NDR, p53, HDM2, and HDM4 binding to human S100BNovel interactions of the TRTK12 peptide with S100 protein family members: specificity and thermodynamic characterization.The Calcium-Dependent Interaction of S100B with Its Protein Targets.The design and delivery of a PKA inhibitory polypeptide to treat SCA1.X-ray crystal structure of human calcium-bound S100A1.
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P2860
The Effects of CapZ Peptide (TRTK-12) Binding to S100B–Ca2+ as Examined by NMR and X-ray Crystallography
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2010 nî lūn-bûn
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2010 թուականի Մարտին հրատարակուած գիտական յօդուած
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2010 թվականի մարտին հրատարակված գիտական հոդված
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2010年の論文
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2010年論文
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2010年論文
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2010年論文
@zh-hk
2010年論文
@zh-mo
2010年論文
@zh-tw
2010年论文
@wuu
name
The Effects of CapZ Peptide (T ...... NMR and X-ray Crystallography
@ast
The Effects of CapZ Peptide (T ...... NMR and X-ray Crystallography
@en
The Effects of CapZ Peptide (T ...... NMR and X-ray Crystallography
@nl
type
label
The Effects of CapZ Peptide (T ...... NMR and X-ray Crystallography
@ast
The Effects of CapZ Peptide (T ...... NMR and X-ray Crystallography
@en
The Effects of CapZ Peptide (T ...... NMR and X-ray Crystallography
@nl
prefLabel
The Effects of CapZ Peptide (T ...... NMR and X-ray Crystallography
@ast
The Effects of CapZ Peptide (T ...... NMR and X-ray Crystallography
@en
The Effects of CapZ Peptide (T ...... NMR and X-ray Crystallography
@nl
P2093
P2860
P3181
P1476
The Effects of CapZ Peptide (T ...... NMR and X-ray Crystallography
@en
P2093
David J Weber
Eric A Toth
Kristen M Varney
Laura E Thompson
Melissa A Liriano
Paul T Wilder
Thomas H Charpentier
P2860
P304
P3181
P356
10.1016/J.JMB.2009.12.057
P407
P577
2010-03-12T00:00:00Z