Correlating AMPA Receptor Activation and Cleft Closure across Subunits: Crystal Structures of the GluR4 Ligand-Binding Domain in Complex with Full and Partial Agonists †
about
Piracetam defines a new binding site for allosteric modulators of alpha-amino-3-hydroxy-5-methyl-4-isoxazole-propionic acid (AMPA) receptorsFunctional insights from glutamate receptor ion channel structuresEnhanced Efficacy without Further Cleft Closure: Reevaluating Twist as a Source of Agonist Efficacy in AMPA ReceptorsMolecular Mechanism of Flop Selectivity and Subsite Recognition for an AMPA Receptor Allosteric Modulator: Structures of GluA2 and GluA3 in Complexes with PEPAMechanism of AMPA Receptor Activation by Partial Agonists: DISULFIDE TRAPPING OF CLOSED LOBE CONFORMATIONSThe Structure of (-)-Kaitocephalin Bound to the Ligand Binding Domain of the (S)- -Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA)/Glutamate Receptor, GluA2The Loss of an Electrostatic Contact Unique to AMPA Receptor Ligand Binding Domain 2 Slows Channel ActivationThermodynamics and Mechanism of the Interaction of Willardiine Partial Agonists with a Glutamate Receptor: Implications for Drug DevelopmentGlutamate receptor ion channels: structure, regulation, and functionDomain architecture of a calcium-permeable AMPA receptor in a ligand-free conformation.Hydrophobic side chain dynamics of a glutamate receptor ligand binding domainRole of dimer interface in activation and desensitization in AMPA receptorsRole of cross-cleft contacts in NMDA receptor gatingDiscovery of a new class of ionotropic glutamate receptor antagonists by the rational design of (2S,3R)-3-(3-carboxyphenyl)-pyrrolidine-2-carboxylic acidStructure and mechanism of glutamate receptor ion channel assembly, activation and modulation.
P2860
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P2860
Correlating AMPA Receptor Activation and Cleft Closure across Subunits: Crystal Structures of the GluR4 Ligand-Binding Domain in Complex with Full and Partial Agonists †
description
2008 nî lūn-bûn
@nan
2008 թուականի Դեկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2008 թվականի դեկտեմբերին հրատարակված գիտական հոդված
@hy
2008年の論文
@ja
2008年論文
@yue
2008年論文
@zh-hant
2008年論文
@zh-hk
2008年論文
@zh-mo
2008年論文
@zh-tw
2008年论文
@wuu
name
Correlating AMPA Receptor Acti ...... th Full and Partial Agonists †
@ast
Correlating AMPA Receptor Acti ...... th Full and Partial Agonists †
@en
Correlating AMPA Receptor Acti ...... th Full and Partial Agonists †
@nl
type
label
Correlating AMPA Receptor Acti ...... th Full and Partial Agonists †
@ast
Correlating AMPA Receptor Acti ...... th Full and Partial Agonists †
@en
Correlating AMPA Receptor Acti ...... th Full and Partial Agonists †
@nl
prefLabel
Correlating AMPA Receptor Acti ...... th Full and Partial Agonists †
@ast
Correlating AMPA Receptor Acti ...... th Full and Partial Agonists †
@en
Correlating AMPA Receptor Acti ...... th Full and Partial Agonists †
@nl
P2093
P2860
P356
P1433
P1476
Correlating AMPA Receptor Acti ...... th Full and Partial Agonists †
@en
P2093
Avinash Gill
Brian L Jones
Dean R Madden
Leslie P Henderson
P2860
P304
P356
10.1021/BI8013196
P407
P577
2008-12-30T00:00:00Z