A combined spectroscopic and crystallographic approach to probing drug-human serum albumin interactions
about
Structural studies of bovine, equine, and leporine serum albumin complexes with naproxenStructural evidence of the species-dependent albumin binding of the modified cyclic phosphatidic acid with cytotoxic propertiesInterpreting physicochemical experimental data sets.11β-Hydroxysteroid dehydrogenase type 1 (11β-HSD1) inhibitors still improve metabolic phenotype in male 11β-HSD1 knockout mice suggesting off-target mechanisms.In silico prediction of human serum albumin binding for drug leads.Potent and selective bivalent inhibitors of BET bromodomains.Continuous inhibition of 11β-hydroxysteroid dehydrogenase type I in adipose tissue leads to tachyphylaxis in humans and rats but not in mice.Domain-specific interactions between MLN8237 and human serum albumin estimated by STD and WaterLOGSY NMR, ITC, spectroscopic, and docking techniques.Interactive association of drugs binding to human serum albumin.Intrinsically Disordered Regions in Serum Albumin: What Are They For?Characterization of the binding sites of the anticancer ruthenium(III) complexes KP1019 and KP1339 on human serum albumin via competition studies.Enantiomeric pairs reveal that key medicinal chemistry parameters vary more than simple physical property based models can explain
P2860
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P2860
A combined spectroscopic and crystallographic approach to probing drug-human serum albumin interactions
description
2010 nî lūn-bûn
@nan
2010 թուականի Նոյեմբերին հրատարակուած գիտական յօդուած
@hyw
2010 թվականի նոյեմբերին հրատարակված գիտական հոդված
@hy
2010年の論文
@ja
2010年学术文章
@wuu
2010年学术文章
@zh-cn
2010年学术文章
@zh-hans
2010年学术文章
@zh-my
2010年学术文章
@zh-sg
2010年學術文章
@yue
name
A combined spectroscopic and c ...... man serum albumin interactions
@ast
A combined spectroscopic and c ...... man serum albumin interactions
@en
A combined spectroscopic and c ...... man serum albumin interactions
@nl
type
label
A combined spectroscopic and c ...... man serum albumin interactions
@ast
A combined spectroscopic and c ...... man serum albumin interactions
@en
A combined spectroscopic and c ...... man serum albumin interactions
@nl
prefLabel
A combined spectroscopic and c ...... man serum albumin interactions
@ast
A combined spectroscopic and c ...... man serum albumin interactions
@en
A combined spectroscopic and c ...... man serum albumin interactions
@nl
P2093
P3181
P1476
A combined spectroscopic and c ...... man serum albumin interactions
@en
P2093
Alleyn Plowright
David Buttar
Holger Steuber
Nicola Colclough
Paul Whittamore
Philip A MacFaul
Scott D Phillips
Stefan Gerhardt
P304
P3181
P356
10.1016/J.BMC.2010.08.052
P407
P577
2010-11-01T00:00:00Z