Design and Synthesis of Inhibitors of Plasmodium falciparumN -Myristoyltransferase, A Promising Target for Antimalarial Drug Discovery
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Structure and Functional Diversity of GCN5-Related N-Acetyltransferases (GNAT)Discovery of Novel and Ligand-Efficient Inhibitors of Plasmodium falciparum and Plasmodium vivax N -MyristoyltransferaseDesign and Synthesis of High Affinity Inhibitors of Plasmodium falciparum and Plasmodium vivax N -Myristoyltransferases Directed by Ligand Efficiency Dependent Lipophilicity (LELP)Diverse modes of binding in structures ofLeishmania majorN-myristoyltransferase with selective inhibitorsStructure of N-myristoyltransferase from Aspergillus fumigatusUnique apicomplexan IMC sub-compartment proteins are early markers for apical polarity in the malaria parasiteAn improved method and cost effective strategy for soluble expression and purification of human N-myristoyltransferase 1 in E. coli.N-myristoyltransferase is a cell wall target in Aspergillus fumigatus.Integrated machine learning, molecular docking and 3D-QSAR based approach for identification of potential inhibitors of trypanosomal N-myristoyltransferase.Discovery of high affinity inhibitors of Leishmania donovani N-myristoyltransferase.Discovery of pyridyl-based inhibitors of Plasmodium falciparum N-myristoyltransferaseRepurposing strategies for tropical disease drug discovery.Chemical proteomics: a powerful tool for exploring protein lipidation.N-Myristoyltransferase as a potential drug target in malaria and leishmaniasis.From crystal to compound: structure-based antimalarial drug discovery.N-Myristoyltransferase Inhibition Induces ER-Stress, Cell Cycle Arrest, and Apoptosis in Cancer Cells.Drug target identification in protozoan parasites.Recent advances in the discovery of N-myristoyltransferase inhibitors.New developments in probing and targeting protein acylation in malaria, leishmaniasis and African sleeping sickness.Stacking with No Planarity?Structure-guided optimization of quinoline inhibitors of Plasmodium N-myristoyltransferase.Structure-based design of potent and selective Leishmania N-myristoyltransferase inhibitors.Design and Synthesis of Brain Penetrant Trypanocidal N-Myristoyltransferase Inhibitors.
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P2860
Design and Synthesis of Inhibitors of Plasmodium falciparumN -Myristoyltransferase, A Promising Target for Antimalarial Drug Discovery
description
2012 nî lūn-bûn
@nan
2012 թուականի Հոկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2012 թվականի հոտեմբերին հրատարակված գիտական հոդված
@hy
2012年の論文
@ja
2012年論文
@yue
2012年論文
@zh-hant
2012年論文
@zh-hk
2012年論文
@zh-mo
2012年論文
@zh-tw
2012年论文
@wuu
name
Design and Synthesis of Inhibi ...... or Antimalarial Drug Discovery
@ast
Design and Synthesis of Inhibi ...... or Antimalarial Drug Discovery
@en
Design and Synthesis of Inhibi ...... or Antimalarial Drug Discovery
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type
label
Design and Synthesis of Inhibi ...... or Antimalarial Drug Discovery
@ast
Design and Synthesis of Inhibi ...... or Antimalarial Drug Discovery
@en
Design and Synthesis of Inhibi ...... or Antimalarial Drug Discovery
@nl
prefLabel
Design and Synthesis of Inhibi ...... or Antimalarial Drug Discovery
@ast
Design and Synthesis of Inhibi ...... or Antimalarial Drug Discovery
@en
Design and Synthesis of Inhibi ...... or Antimalarial Drug Discovery
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P2860
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P921
P3181
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P1476
Design and Synthesis of Inhibi ...... or Antimalarial Drug Discovery
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P2093
A Marek Brzozowski
David K Moss
James A Brannigan
Robin J Leatherbarrow
Zhiyong Yu
P2860
P304
P3181
P356
10.1021/JM301160H
P407
P577
2012-10-25T00:00:00Z