Design and synthesis of conformationally constrained inhibitors of non-nucleoside reverse transcriptase
about
Antiviral activity and in vitro mutation development pathways of MK-6186, a novel nonnucleoside reverse transcriptase inhibitorAllosteric modulation of protein oligomerization: an emerging approach to drug design.Conformational restriction: an effective tactic in 'follow-on'-based drug discovery.Design, synthesis, and biological evaluation of novel trifluoromethyl indoles as potent HIV-1 NNRTIs with an improved drug resistance profile.3-substituted indazoles as configurationally locked 4EGI-1 mimetics and inhibitors of the eIF4E/eIF4G interaction.Biological activity of sporolides A and B from Salinispora tropica: in silico target prediction using ligand-based pharmacophore mapping and in vitro activity validation on HIV-1 reverse transcriptase.
P2860
Design and synthesis of conformationally constrained inhibitors of non-nucleoside reverse transcriptase
description
2011 nî lūn-bûn
@nan
2011 թուականի Նոյեմբերին հրատարակուած գիտական յօդուած
@hyw
2011 թվականի նոյեմբերին հրատարակված գիտական հոդված
@hy
2011年の論文
@ja
2011年論文
@yue
2011年論文
@zh-hant
2011年論文
@zh-hk
2011年論文
@zh-mo
2011年論文
@zh-tw
2011年论文
@wuu
name
Design and synthesis of confor ...... cleoside reverse transcriptase
@ast
Design and synthesis of confor ...... cleoside reverse transcriptase
@en
Design and synthesis of confor ...... cleoside reverse transcriptase
@nl
type
label
Design and synthesis of confor ...... cleoside reverse transcriptase
@ast
Design and synthesis of confor ...... cleoside reverse transcriptase
@en
Design and synthesis of confor ...... cleoside reverse transcriptase
@nl
prefLabel
Design and synthesis of confor ...... cleoside reverse transcriptase
@ast
Design and synthesis of confor ...... cleoside reverse transcriptase
@en
Design and synthesis of confor ...... cleoside reverse transcriptase
@nl
P2093
P356
P1476
Design and synthesis of confor ...... cleoside reverse transcriptase
@en
P2093
Bang-Lin Wan
Brenda Paton
Daniel Distefano
Georgia McGaughey
Jessica Flynn
Joseph P Vacca
Maricel Torrent
Mike Miller
Ming-Tain Lai
P304
P356
10.1021/JM2010173
P407
P577
2011-11-24T00:00:00Z