Systematic comparison of peptidic proteasome inhibitors highlights the α-ketoamide electrophile as an auspicious reversible lead motif

Systematic comparison of peptidic proteasome inhibitors highlights the α-ketoamide electrophile as an auspicious reversible lead motif

Item
http://www.wikidata.org/entity/Q27688108
α-Keto phenylamides as P1'-extended proteasome inhibitorsSelective inhibition of the immunoproteasome by ligand-induced crosslinking of the active siteIndolo-phakellins as β5-specific noncovalent proteasome inhibitorsA Minimal β-Lactone Fragment for Selective β5c or β5i Proteasome InhibitorsTargeted Delivery of Proteasome Inhibitors to Somatostatin-Receptor-Expressing Cancer Cells by Octreotide ConjugationA unified mechanism for proteolysis and autocatalytic activation in the 20S proteasome.Synthesis, bioactivity, docking and molecular dynamics studies of furan-based peptides as 20S proteasome inhibitors.Development of novel selective peptidomimetics containing a boronic acid moiety, targeting the 20S proteasome as anticancer agents.Rational Design of Proteasome Inhibitors as Antimalarial Drugs.Cryo-EM reveals the conformation of a substrate analogue in the human 20S proteasome core.Tunable Probes with Direct Fluorescence Signals for the Constitutive and Immunoproteasome.Structural Elucidation of a Nonpeptidic Inhibitor Specific for the Human Immunoproteasome.One pot synthesis of α-ketoamides from ethylarenes and amines: a metal free difunctionalization strategy.Unbiased compound-protein interface mapping and prediction of chemoresistance loci through forward genetics in haploid stem cells.Visible-light initiated copper(i)-catalysed oxidative C–N coupling of anilines with terminal alkynes: one-step synthesis of α-ketoamides
P2860

Systematic comparison of peptidic proteasome inhibitors highlights the α-ketoamide electrophile as an auspicious reversible lead motif

Item
http://www.wikidata.org/entity/Q27688108
description
2014 nî lūn-bûn
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2014 թուականի Փետրուարին հրատարակուած գիտական յօդուած
@hyw
2014 թվականի փետրվարին հրատարակված գիտական հոդված
@hy
2014年の論文
@ja
2014年論文
@yue
2014年論文
@zh-hant
2014年論文
@zh-hk
2014年論文
@zh-mo
2014年論文
@zh-tw
2014年论文
@wuu
name
Systematic comparison of pepti ...... spicious reversible lead motif
@ast
Systematic comparison of pepti ...... spicious reversible lead motif
@en
Systematic comparison of pepti ...... spicious reversible lead motif
@nl
type
label
Systematic comparison of pepti ...... spicious reversible lead motif
@ast
Systematic comparison of pepti ...... spicious reversible lead motif
@en
Systematic comparison of pepti ...... spicious reversible lead motif
@nl
prefLabel
Systematic comparison of pepti ...... spicious reversible lead motif
@ast
Systematic comparison of pepti ...... spicious reversible lead motif
@en
Systematic comparison of pepti ...... spicious reversible lead motif
@nl
P1433
P1476
P2093
P2860
P304
P31
P356
P407
P433
P478
P50
P577
P698
P356
P1433
P1476
Systematic comparison of pepti ...... spicious reversible lead motif
@en
P2093
P2860
P304
P31
P356
P407
P433
P478
P50
P577
P698