Conformation-Selective Analogues of Dasatinib Reveal Insight into Kinase Inhibitor Binding and Selectivity
about
Structural and Biochemical Basis for Intracellular Kinase Inhibition by Src-specific Peptidic MacrocyclesThe impact of Thr91 mutation on c-Src resistance to UM-164: molecular dynamics study revealed a new opportunity for drug design.Conquering the challenges of genotypic and phenotypic tumor heterogeneity to realize the promise of personalized cancer therapy: the role of academia.How and when does an anticancer drug leave its binding site?Emergence of a Promising Lead Compound in the Treatment of Triple Negative Breast Cancer: An Insight into Conformational Features and Ligand Binding Landscape of c-Src Protein with UM-164.Survey of solution dynamics in Src kinase reveals allosteric cross talk between the ligand binding and regulatory sites.Activation loop targeting strategy for design of receptor-interacting protein kinase 2 (RIPK2) inhibitors.
P2860
Q27727987-6A0A0B3D-EC75-4A55-B14F-71460234142CQ30401596-707A2078-6DA6-492D-BC36-6CDF42ED46A3Q41112169-B050BB67-E62C-4925-9E0C-CE038A50F94DQ41965081-070F0E33-41F0-4D18-A1E0-47020FFAF6B5Q47250599-6C3B6421-A1AD-46EB-AF51-D34B4E68FDCDQ47279026-9FC6A389-67AE-4C08-B4F4-472AEE7854F2Q48509895-261DC45F-98F4-4448-85D9-4B92C2D63405
P2860
Conformation-Selective Analogues of Dasatinib Reveal Insight into Kinase Inhibitor Binding and Selectivity
description
2016 nî lūn-bûn
@nan
2016 թուականի Մայիսին հրատարակուած գիտական յօդուած
@hyw
2016 թվականի մայիսին հրատարակված գիտական հոդված
@hy
2016年の論文
@ja
2016年論文
@yue
2016年論文
@zh-hant
2016年論文
@zh-hk
2016年論文
@zh-mo
2016年論文
@zh-tw
2016年论文
@wuu
name
Conformation-Selective Analogu ...... ibitor Binding and Selectivity
@ast
Conformation-Selective Analogu ...... ibitor Binding and Selectivity
@en
Conformation-Selective Analogu ...... ibitor Binding and Selectivity
@nl
type
label
Conformation-Selective Analogu ...... ibitor Binding and Selectivity
@ast
Conformation-Selective Analogu ...... ibitor Binding and Selectivity
@en
Conformation-Selective Analogu ...... ibitor Binding and Selectivity
@nl
prefLabel
Conformation-Selective Analogu ...... ibitor Binding and Selectivity
@ast
Conformation-Selective Analogu ...... ibitor Binding and Selectivity
@en
Conformation-Selective Analogu ...... ibitor Binding and Selectivity
@nl
P2093
P1433
P1476
Conformation-Selective Analogu ...... ibitor Binding and Selectivity
@en
P2093
Frank E Kwarcinski
Jeanne A Stuckey
Jennifer L Meagher
Kristoffer R Brandvold
Matthew B Soellner
Omar M Beleh
Sameer Phadke
Taylor K Johnson
P304
P356
10.1021/ACSCHEMBIO.5B01018
P577
2016-03-01T00:00:00Z