Serine protease mechanism: structure of an inhibitory complex of alpha-lytic protease and a tightly bound peptide boronic acid
about
Three decades of beta-lactamase inhibitorsAtomic resolution structure of a lysine-specific endoproteinase from Lysobacter enzymogenes suggests a hydroxyl group bound to the oxyanion holeStructure of alpha-lytic protease complexed with its pro regionEnzyme specificity under dynamic control II: Principal component analysis of alpha-lytic protease using global and local solvent boundary conditionsStructural basis of substrate specificity in the serine proteasesRecent developments in inhibiting cysteine and serine proteases.Repurposing Suzuki Coupling Reagents as a Directed Fragment Library Targeting Serine Hydrolases and Related EnzymesPentapeptide boronic acid inhibitors of Mycobacterium tuberculosis MycP1 protease.Crystal versus solution structure of enzymes: NMR spectroscopy of a peptide boronic acid-serine protease complex in the crystalline stateDiscovery of 2-[5-(4-Fluorophenylcarbamoyl)pyridin-2-ylsulfanylmethyl]phenylboronic Acid (SX-517): Noncompetitive Boronic Acid Antagonist of CXCR1 and CXCR2Cytotoxic and apoptotic effects of boron compounds on leukemia cell line.Cellular changes in boric acid-treated DU-145 prostate cancer cells.Assembly of an active enzyme by the linkage of two protein modules.Analysis of prepro-alpha-lytic protease expression in Escherichia coli reveals that the pro region is required for activityConformational substates in enzyme mechanism: the 120 K structure of alpha-lytic protease at 1.5 A resolution.Peptide and Peptide-Like Modulators of 20S Proteasome Enzymatic Activity in Cancer CellsHollow boron nitride nanospheres as boron reservoir for prostate cancer treatment.Prostate-specific antigen: an overlooked candidate for the targeted treatment and selective imaging of prostate cancer.A 13C-NMR study of the role of Asn-155 in stabilizing the oxyanion of a subtilisin tetrahedral adduct.Potent and selective peptidyl boronic acid inhibitors of the serine protease prostate-specific antigen.Benzyloxycarbonyl-D-Phe-Pro-methoxypropylboroglycine: a novel inhibitor of thrombin with high selectivity containing a neutral side chain at the P1 position.Correct folding of alpha-lytic protease is required for its extracellular secretion from Escherichia coli.Slow tight binding inhibition of proteinase K by a proteinaceous inhibitor: conformational alterations responsible for conferring irreversibility to the enzyme-inhibitor complex.The apoptotic, cytotoxic and genotoxic effect of novel binuclear boron-fluoride complex on endometrial cancer.Boric acid-dependent decrease in regulatory histone H3 acetylation is not mutagenic in yeast.Direct evidence of a low barrier hydrogen bond in the catalytic triad of a Serine proteaseStructural Analyses on Intermediates in Serine Protease Catalysis
P2860
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P2860
Serine protease mechanism: structure of an inhibitory complex of alpha-lytic protease and a tightly bound peptide boronic acid
description
1987 nî lūn-bûn
@nan
1987 թուականի Դեկտեմբերին հրատարակուած գիտական յօդուած
@hyw
1987 թվականի դեկտեմբերին հրատարակված գիտական հոդված
@hy
1987年の論文
@ja
1987年学术文章
@wuu
1987年学术文章
@zh-cn
1987年学术文章
@zh-hans
1987年学术文章
@zh-my
1987年学术文章
@zh-sg
1987年學術文章
@yue
name
Serine protease mechanism: str ...... tly bound peptide boronic acid
@ast
Serine protease mechanism: str ...... tly bound peptide boronic acid
@en
Serine protease mechanism: str ...... tly bound peptide boronic acid
@nl
type
label
Serine protease mechanism: str ...... tly bound peptide boronic acid
@ast
Serine protease mechanism: str ...... tly bound peptide boronic acid
@en
Serine protease mechanism: str ...... tly bound peptide boronic acid
@nl
prefLabel
Serine protease mechanism: str ...... tly bound peptide boronic acid
@ast
Serine protease mechanism: str ...... tly bound peptide boronic acid
@en
Serine protease mechanism: str ...... tly bound peptide boronic acid
@nl
P2093
P356
P1433
P1476
Serine protease mechanism: str ...... tly bound peptide boronic acid
@en
P2093
P304
P356
10.1021/BI00398A012
P407
P577
1987-12-01T00:00:00Z