Functionally selective dopamine D₂, D₃ receptor partial agonists
about
Structure-based discovery of opioid analgesics with reduced side effects.Dopamine receptors - IUPHAR Review 13Receptor, Ligand and Transducer Contributions to Dopamine D2 Receptor Functional Selectivity.Comparative MD Simulations Indicate a Dual Role for Arg1323.50 in Dopamine-Dependent D2R Activation.Identifying Medication Targets for Psychostimulant Addiction: Unraveling the Dopamine D3 Receptor Hypothesis.The role of kinetic context in apparent biased agonism at GPCRs.Efficacy of Hybrid Tetrahydrobenzo[d]thiazole Based Aryl Piperazines D-264 and D-301 at D₂ and D₃ ReceptorsMultivalent approaches and beyond: novel tools for the investigation of dopamine D2 receptor pharmacology.Functional selectivity at G-protein coupled receptors: Advancing cannabinoid receptors as drug targets.Novel Molecular Strategies and Targets for Opioid Drug Discovery for the Treatment of Chronic Pain.Discovery of novel brain permeable and G protein-biased beta-1 adrenergic receptor partial agonists for the treatment of neurocognitive disorders.Synthesis, Molecular Properties Estimations, and Dual Dopamine D2 and D3 Receptor Activities of Benzothiazole-Based Ligands.New approach toward the synthesis of deuterated pyrazolo[1,5-a]pyridines and 1,2,4-triazolo[1,5-a]pyridines.Structure-based evolution of subtype-selective neurotensin receptor ligands.Discovery of G Protein-Biased D2 Dopamine Receptor Partial Agonists.Bioluminescence Resonance Energy Transfer Assay to Characterize Gi-Like G Protein Subtype-Dependent Functional Selectivity.Photochromic Dopamine Receptor Ligands Based on Dithienylethenes and Fulgides.Synthesis, Biological, and Computational Evaluation of Substituted 1-(2-Methoxyphenyl)-4-(1-phenethylpiperidin-4-yl)piperazines and 1-(2-Methoxyphenyl)-4-[(1-phenethylpiperidin-4-yl)methyl]piperazines as Dopaminergic Ligands.Structure-Activity Investigation of a G Protein-Biased Agonist Reveals Molecular Determinants for Biased Signaling of the D2 Dopamine Receptor.
P2860
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P2860
Functionally selective dopamine D₂, D₃ receptor partial agonists
description
2014 nî lūn-bûn
@nan
2014 թուականի Յունիսին հրատարակուած գիտական յօդուած
@hyw
2014 թվականի հունիսին հրատարակված գիտական հոդված
@hy
2014年の論文
@ja
2014年論文
@yue
2014年論文
@zh-hant
2014年論文
@zh-hk
2014年論文
@zh-mo
2014年論文
@zh-tw
2014年论文
@wuu
name
Functionally selective dopamine D₂, D₃ receptor partial agonists
@ast
Functionally selective dopamine D₂, D₃ receptor partial agonists
@en
Functionally selective dopamine D₂, D₃ receptor partial agonists
@nl
type
label
Functionally selective dopamine D₂, D₃ receptor partial agonists
@ast
Functionally selective dopamine D₂, D₃ receptor partial agonists
@en
Functionally selective dopamine D₂, D₃ receptor partial agonists
@nl
prefLabel
Functionally selective dopamine D₂, D₃ receptor partial agonists
@ast
Functionally selective dopamine D₂, D₃ receptor partial agonists
@en
Functionally selective dopamine D₂, D₃ receptor partial agonists
@nl
P2093
P356
P1476
Functionally selective dopamine D₂, D₃ receptor partial agonists
@en
P2093
Dorothee Möller
Harald Hübner
Kristina Leuner
Marika Skultety
Ralf C Kling
P304
P356
10.1021/JM5004039
P407
P577
2014-06-12T00:00:00Z