Cocaine and 3 beta-(4'-substituted phenyl)tropane-2 beta-carboxylic acid ester and amide analogues. New high-affinity and selective compounds for the dopamine transporter
about
Positive allosteric modulation of the human cannabinoid (CB) receptor by RTI-371, a selective inhibitor of the dopamine transporterKappa opioids as potential treatments for stimulant dependenceMultiple ADH genes modulate risk for drug dependence in both African- and European-AmericansImaging the serotonin transporter during major depressive disorder and antidepressant treatmentFaster onset and dopamine transporter selectivity predict stimulant and reinforcing effects of cocaine analogs in squirrel monkeysSynthesis, fluorine-18 radiolabeling, and biological evaluation of N-((E)-4-fluorobut-2-en-1-yl)-2beta-carbomethoxy-3beta-(4'-halophenyl)nortropanes: candidate radioligands for in vivo imaging of the brain dopamine transporter with positron emissionDevelopment of 3-phenyltropane analogues with high affinity for the dopamine and serotonin transporters and low affinity for the norepinephrine transporter.[(125)I]3beta-(4-ethyl-3-iodophenyl)nortropane-2beta-carboxylic acid methyl ester ([(125)I]EINT): a potent and selective radioligand for the brain serotonin transporter.Self-administration of cocaine and the cocaine analog RTI-113: relationship to dopamine transporter occupancy determined by PET neuroimaging in rhesus monkeys.Probes for the dopamine transporter: new leads toward a cocaine-abuse therapeutic--A focus on analogues of benztropine and rimcazole.Interaction of tyrosine 151 in norepinephrine transporter with the 2β group of cocaine analog RTI-113.Self-administration of drug mixtures by monkeys: combining drugs with comparable mechanisms of actionNicotinic acetylcholine receptor efficacy and pharmacological properties of 3-(substituted phenyl)-2β-substituted tropanes.The novel trisubstituted pyran derivative D-142 has triple monoamine reuptake inhibitory activity and exerts potent antidepressant-like activity in rodents.Pharmacophore-based discovery of ligands for drug transporters.Synthesis and evaluation of novel tropane derivatives as potential PET imaging agents for the dopamine transporter.Voltammetric characterization of the effect of monoamine uptake inhibitors and releasers on dopamine and serotonin uptake in mouse caudate-putamen and substantia nigra slices.The solute carrier 6 family of transportersThe synthesis of bivalent 2beta-carbomethoxy-3beta-(3,4-dichlorophenyl)-8-heterobicyclo[3.2.1]octanes as probes for proximal binding sites on the dopamine and serotonin transporters.Depletion of serotonin decreases the effects of the kappa-opioid receptor agonist U-69593 on cocaine-stimulated activitySynthesis, radiosynthesis, and biological evaluation of fluorine-18-labeled 2beta-carbo(fluoroalkoxy)-3beta-(3'-((Z)-2-haloethenyl)phenyl)nortropanes: candidate radioligands for in vivo imaging of the serotonin transporter with positron emission tomFluorine-18 Radiolabeled PET Tracers for Imaging Monoamine Transporters: Dopamine, Serotonin, and Norepinephrine.Biophysical characterization of the cocaine binding pocket in the serotonin transporter using a fluorescent cocaine analogue as a molecular reporter.Chronic cocaine increases kappa-opioid receptor density: lack of effect by selective dopamine uptake inhibitors.Demonstration of clomipramine and venlafaxine occupation at serotonin reuptake sites in man in vivo.
P2860
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P2860
Cocaine and 3 beta-(4'-substituted phenyl)tropane-2 beta-carboxylic acid ester and amide analogues. New high-affinity and selective compounds for the dopamine transporter
description
1995 nî lūn-bûn
@nan
1995 թուականի Յունուարին հրատարակուած գիտական յօդուած
@hyw
1995 թվականի հունվարին հրատարակված գիտական հոդված
@hy
1995年の論文
@ja
1995年論文
@yue
1995年論文
@zh-hant
1995年論文
@zh-hk
1995年論文
@zh-mo
1995年論文
@zh-tw
1995年论文
@wuu
name
Cocaine and 3 beta-(4'-substit ...... s for the dopamine transporter
@ast
Cocaine and 3 beta-(4'-substit ...... s for the dopamine transporter
@en
Cocaine and 3 beta-(4'-substit ...... s for the dopamine transporter
@nl
type
label
Cocaine and 3 beta-(4'-substit ...... s for the dopamine transporter
@ast
Cocaine and 3 beta-(4'-substit ...... s for the dopamine transporter
@en
Cocaine and 3 beta-(4'-substit ...... s for the dopamine transporter
@nl
prefLabel
Cocaine and 3 beta-(4'-substit ...... s for the dopamine transporter
@ast
Cocaine and 3 beta-(4'-substit ...... s for the dopamine transporter
@en
Cocaine and 3 beta-(4'-substit ...... s for the dopamine transporter
@nl
P2093
P356
P1476
Cocaine and 3 beta-(4'-substit ...... s for the dopamine transporter
@en
P2093
A Dehghani
F I Carroll
K A Parham
M A Kuzemko
P304
P356
10.1021/JM00002A020
P407
P577
1995-01-20T00:00:00Z