KNI-102, a novel tripeptide HIV protease inhibitor containing allophenylnorstatine as a transition-state mimic
about
Crystal Structures of the Histo-Aspartic Protease (HAP) from Plasmodium falciparumCrystal structures of the free and inhibited forms of plasmepsin I (PMI) from Plasmodium falciparumStructural Insights into the Activation and Inhibition of Histo-Aspartic Protease from Plasmodium falciparumCrystal structures of multidrug-resistant HIV-1 protease in complex with two potent anti-malarial compoundsIn vitro anti-human immunodeficiency virus (HIV) activities of transition state mimetic HIV protease inhibitors containing allophenylnorstatineAntimalarial activity enhancement in hydroxymethylcarbonyl (HMC) isostere-based dipeptidomimetics targeting malarial aspartic protease plasmepsin.Understanding the structural basis of substrate recognition by Plasmodium falciparum plasmepsin V to aid in the design of potent inhibitors.Design of potent aspartic protease inhibitors to treat various diseases.The application of bioisosteres in drug design for novel drug discovery: focusing on acid protease inhibitors.Design and synthesis of substrate-based peptidomimetic human immunodeficiency virus protease inhibitors containing the hydroxymethylcarbonyl isostere.Search for substrate-based inhibitors fitting the S2' space of malarial aspartic protease plasmepsin II.
P2860
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P2860
KNI-102, a novel tripeptide HIV protease inhibitor containing allophenylnorstatine as a transition-state mimic
description
1991 nî lūn-bûn
@nan
1991 թուականի Նոյեմբերին հրատարակուած գիտական յօդուած
@hyw
1991 թվականի նոյեմբերին հրատարակված գիտական հոդված
@hy
1991年の論文
@ja
1991年論文
@yue
1991年論文
@zh-hant
1991年論文
@zh-hk
1991年論文
@zh-mo
1991年論文
@zh-tw
1991年论文
@wuu
name
KNI-102, a novel tripeptide HI ...... ne as a transition-state mimic
@ast
KNI-102, a novel tripeptide HI ...... ne as a transition-state mimic
@en
KNI-102, a novel tripeptide HI ...... ne as a transition-state mimic
@nl
type
label
KNI-102, a novel tripeptide HI ...... ne as a transition-state mimic
@ast
KNI-102, a novel tripeptide HI ...... ne as a transition-state mimic
@en
KNI-102, a novel tripeptide HI ...... ne as a transition-state mimic
@nl
prefLabel
KNI-102, a novel tripeptide HI ...... ne as a transition-state mimic
@ast
KNI-102, a novel tripeptide HI ...... ne as a transition-state mimic
@en
KNI-102, a novel tripeptide HI ...... ne as a transition-state mimic
@nl
P2093
P3181
P356
P1476
KNI-102, a novel tripeptide HI ...... ne as a transition-state mimic
@en
P2093
S Kisanuki
P304
P3181
P356
10.1248/CPB.39.3088
P407
P577
1991-11-01T00:00:00Z