Triterpene derivatives that block entry of human immunodeficiency virus type 1 into cells
about
Sensitivity to a nonpeptidic compound (RPR103611) blocking human immunodeficiency virus type 1 Env-mediated fusion depends on sequence and accessibility of the gp41 loop regionRole of human immunodeficiency virus (HIV) type 1 envelope in the anti-HIV activity of the betulinic acid derivative IC9564Characterization of siamycin I, a human immunodeficiency virus fusion inhibitorResistance to a drug blocking human immunodeficiency virus type 1 entry (RPR103611) is conferred by mutations in gp41Characterization of a novel type of HIV-1 particle assembly inhibitor using a quantitative luciferase-Vpr packaging-based assaySynthesis of antitumor-active betulinic acid-derived hydroxypropargylamines by copper-catalyzend mannich reactions.Synthesis, encapsulation and antitumor activity of new betulin derivatives.Discovery, synthesis, and biological evaluation of a novel group of selective inhibitors of filoviral entryBetulinic acid suppresses constitutive and TNFalpha-induced NF-kappaB activation and induces apoptosis in human prostate carcinoma PC-3 cells.Novel compounds in preclinical/early clinical development for the treatment of HIV infections.A low-molecular-weight entry inhibitor of both CCR5- and CXCR4-tropic strains of human immunodeficiency virus type 1 targets a novel site on gp41Biotransformation of the antimelanoma agent betulinic acid by Bacillus megaterium ATCC 13368.Current lead natural products for the chemotherapy of human immunodeficiency virus (HIV) infection.Ionic derivatives of betulinic acid as novel HIV-1 protease inhibitors.A small-molecule antagonist of virion assembly.HIV entry inhibitors and their potential in HIV therapyNew anti-HIV agents and targets.Antiviral therapy for human immunodeficiency virus infectionsBifunctional anti-human immunodeficiency virus type 1 small molecules with two novel mechanisms of action.Ionic derivatives of betulinic acid exhibit antiviral activity against herpes simplex virus type-2 (HSV-2), but not HIV-1 reverse transcriptaseThe discovery of a class of novel HIV-1 maturation inhibitors and their potential in the therapy of HIV.A mimic of HIV-1 nucleocapsid protein impairs reverse transcription and displays antiviral activity.New betulinic acid derivatives for bevirimat-resistant human immunodeficiency virus type-1.Plant-derived triterpenoids and analogues as antitumor and anti-HIV agentsAnti-AIDS agents. 78. Design, synthesis, metabolic stability assessment, and antiviral evaluation of novel betulinic acid derivatives as potent anti-human immunodeficiency virus (HIV) agentsProteasome regulators: activators and inhibitors.HIV microbicides: state-of-the-art and new perspectives on the development of entry inhibitors.Amphipathic properties of HIV-1 gp41 fusion inhibitors.Escape from human immunodeficiency virus type 1 (HIV-1) entry inhibitors.Betulinic Acid: Recent Advances in Chemical Modifications, Effective Delivery, and Molecular Mechanisms of a Promising Anticancer Therapy.Hyaluronidase Inhibitory Activity of Pentacylic Triterpenoids from Prismatomeris tetrandra (Roxb.) K. Schum: Isolation, Synthesis and QSAR Study.Activation and inhibition of the proteasome by betulinic acid and its derivatives.Role of the ectodomain of the gp41 transmembrane envelope protein of human immunodeficiency virus type 1 in late steps of the membrane fusion process.Oxysterols, but not cholesterol, inhibit human immunodeficiency virus replication in vitro.Tri-N-Boc-tetraazamacrocycle-nucleoside conjugates: synthesis and anti-HIV activities.An amphiphilic conjugate approach toward the design and synthesis of betulinic acid-polyphenol conjugates as inhibitors of the HIV-1 gp41 fusion core formation.Production of a highly potent epoxide through the microbial metabolism of 3β-acetoxyurs-11-en-13β,28-olide by Aspergillus niger culture.A new single-stage method for obtaining of betulin phenylcarbamates.Safety evaluation of a new anxiolytic product containing botanicals Souroubea spp. and Platanus spp. in dogs.Poly(lactic-co-glycolic acid)-loaded nanoparticles of betulinic acid for improved treatment of hepatic cancer: characterization, in vitro and in vivo evaluations.
P2860
Q28343901-D6BEF1C1-AA55-4BE6-921F-55953C421EADQ28345233-3A5CB173-4A62-4806-9096-601679E0C399Q28379084-27F49BFE-1AA2-4C23-B47A-2AD9040683FBQ28379194-5F88EA56-F298-4B60-9109-6F501734C351Q28477791-BB6A980C-12EA-47D5-B675-D7FB1FEEF3DEQ30317883-6372718D-130A-478A-9632-1B96FF64A31CQ30318499-EC64A2CF-7C5C-4FBA-918D-ECD437A3D872Q33785133-8C8FA4C9-B7ED-47BC-A78D-15D3FD6FBFE4Q33830333-73F8F519-DF47-4085-8484-26C8D8F223F6Q33966254-49F890A7-353D-448B-88C5-DC4BFC401A70Q33966639-4EF71CAC-2C05-4BB8-BD47-AFB306D7D0DAQ33987607-280D8DB9-31ED-4A80-8C86-B1B42BAF1670Q33996826-1216E972-7EC0-460E-B1B3-ED38ABF29154Q34045239-2E2267D8-5357-4226-83D7-1FA1F9FDFB10Q34489215-C7D0F8FE-25E3-4D01-909C-18043D84D0D2Q34595921-951437CD-CFFD-43F5-8568-09802A8FA77DQ34944447-DEE1671C-C563-4644-97AE-607F56D669B3Q35366050-6B4A7BCB-BA76-4F73-8080-B53DE0D675FAQ35548195-6C078E15-A3ED-402D-B916-CA7B9BC200AFQ35828340-DF2576AC-4960-47E5-AFC2-2FB4AC8416C4Q36187060-FA02199E-19EB-4A1A-A77D-E9A72CC32D0EQ36332732-3B67D4F2-FCED-4A27-A29A-AB638E0EAFE4Q36691642-D608DEFA-B0DC-4DD1-9FF6-BF00523D95FFQ37173329-D28984CE-6EA4-407C-8DA7-AB633CFE31C1Q37330178-6DF20716-D8C5-45FB-BFD1-331F841308E0Q37411350-B4F2B5A5-A060-47A0-8AD8-6965AC48FE0CQ37855900-886C5335-22F5-4DFA-9C0C-13FBA95D7C51Q37951610-D796D573-27E9-4F58-A3C5-6BFE0557C780Q38076139-32B71E34-C9B7-439D-9DF6-FC69383E6B53Q38624961-09DB0722-ADAC-40AD-98C9-088DC6F22823Q38861625-70203C00-66F5-482E-A7AF-36A47D4D8727Q40074485-B4563DE9-F675-4B40-8B74-F30BC343DE76Q40604377-659CD4F8-C064-47A0-91F4-C7A78612D8AAQ40985917-0E629E6A-5AE4-4847-AA87-B91A0CD6712BQ41015629-C6A871FE-6342-44C0-9628-0303B4932EABQ42732016-7A61E284-0AB7-4FD7-8943-264A9EB9E449Q46614586-0B69561D-1022-428E-A921-FB23307B77A9Q47804153-7168D9BE-0A7E-4CBA-8E1B-B0261BE20BE4Q49570576-1BD3951E-2AEA-4613-AA4C-9F6D709F1AABQ50335864-F99B3F63-4331-4E66-9676-D9AE5EE15A80
P2860
Triterpene derivatives that block entry of human immunodeficiency virus type 1 into cells
description
1994 nî lūn-bûn
@nan
1994 թուականի Ապրիլին հրատարակուած գիտական յօդուած
@hyw
1994 թվականի ապրիլին հրատարակված գիտական հոդված
@hy
1994年の論文
@ja
1994年論文
@yue
1994年論文
@zh-hant
1994年論文
@zh-hk
1994年論文
@zh-mo
1994年論文
@zh-tw
1994年论文
@wuu
name
Triterpene derivatives that block entry of human immunodeficiency virus type 1 into cells
@ast
Triterpene derivatives that block entry of human immunodeficiency virus type 1 into cells
@en
Triterpene derivatives that block entry of human immunodeficiency virus type 1 into cells
@nl
type
label
Triterpene derivatives that block entry of human immunodeficiency virus type 1 into cells
@ast
Triterpene derivatives that block entry of human immunodeficiency virus type 1 into cells
@en
Triterpene derivatives that block entry of human immunodeficiency virus type 1 into cells
@nl
prefLabel
Triterpene derivatives that block entry of human immunodeficiency virus type 1 into cells
@ast
Triterpene derivatives that block entry of human immunodeficiency virus type 1 into cells
@en
Triterpene derivatives that block entry of human immunodeficiency virus type 1 into cells
@nl
P2093
P2860
P356
P1476
Triterpene derivatives that block entry of human immunodeficiency virus type 1 into cells
@en
P2093
A Bousseau
J F Mayaux
P2860
P304
P356
10.1073/PNAS.91.9.3564
P407
P577
1994-04-26T00:00:00Z