Conjugated enynes as nonaromatic catechol bioisosteres: synthesis, binding experiments, and computational studies of novel dopamine receptor agonists recognizing preferentially the D(3) subtype
about
Structure-based discovery of opioid analgesics with reduced side effects.Visualization and ligand-induced modulation of dopamine receptor dimerization at the single molecule level.Covalent agonists for studying G protein-coupled receptor activationStructure-guided development of heterodimer-selective GPCR ligandsA series of 18F-labelled pyridinylphenyl amides as subtype-selective radioligands for the dopamine D3 receptor.In vivo monitoring of the antiangiogenic effect of neurotensin receptor-mediated radiotherapy by small-animal positron emission tomography: a pilot study.Radical arylation of tyrosine and its application in the synthesis of a highly selective neurotensin receptor 2 ligand.Electrostatic potentials and average electron densities of bioisosteres in methylsquarate and acetic acid.Development of a metabolically stable neurotensin receptor 2 (NTS2) ligand.On the terminal homologation of physiologically active peptides as a means of increasing stability in human serum--neurotensin, opiorphin, B27-KK10 epitope, NPY.Engineering a GPCR-ligand pair that simulates the activation of D(2L) by Dopamine.Identification of the Beer Component Hordenine as Food-Derived Dopamine D2 Receptor Agonist by Virtual Screening a 3D Compound DatabaseIodination of carbohydrate-derived 1,2-oxazines to enantiopure 5-iodo-3,6-dihydro-2H-1,2-oxazines and subsequent palladium-catalyzed cross-coupling reactionsStructure-based evolution of subtype-selective neurotensin receptor ligands.Syntheses, receptor bindings, in vitro and in vivo stabilities and biodistributions of DOTA-neurotensin(8-13) derivatives containing β-amino acid residues - a lesson about the importance of animal experiments.Impact of the proline residue on ligand binding of neurotensin receptor 2 (NTS2)-selective peptide-peptoid hybrids.Structure-Based Design and Discovery of New M2 Receptor Agonists.Routes to drug design via bioisosterism of carboxyl and sulfonamide groups.Photochromic Dopamine Receptor Ligands Based on Dithienylethenes and Fulgides.[18F]Fluorophenylazocarboxylates: Design and Synthesis of Potential Radioligands for Dopamine D3 and μ-Opioid Receptor.In silico studies targeting G-protein coupled receptors for drug research against Parkinson's disease.Hydrido-Cobalt Catalyst as a Selective Tool for the Dimerisation of Arylacetylenes: Scope and Theoretical Studies
P2860
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P2860
Conjugated enynes as nonaromatic catechol bioisosteres: synthesis, binding experiments, and computational studies of novel dopamine receptor agonists recognizing preferentially the D(3) subtype
description
2000 nî lūn-bûn
@nan
2000 թուականի Փետրուարին հրատարակուած գիտական յօդուած
@hyw
2000 թվականի փետրվարին հրատարակված գիտական հոդված
@hy
2000年の論文
@ja
2000年論文
@yue
2000年論文
@zh-hant
2000年論文
@zh-hk
2000年論文
@zh-mo
2000年論文
@zh-tw
2000年论文
@wuu
name
Conjugated enynes as nonaromat ...... referentially the D(3) subtype
@ast
Conjugated enynes as nonaromat ...... referentially the D(3) subtype
@en
Conjugated enynes as nonaromat ...... referentially the D(3) subtype
@nl
type
label
Conjugated enynes as nonaromat ...... referentially the D(3) subtype
@ast
Conjugated enynes as nonaromat ...... referentially the D(3) subtype
@en
Conjugated enynes as nonaromat ...... referentially the D(3) subtype
@nl
prefLabel
Conjugated enynes as nonaromat ...... referentially the D(3) subtype
@ast
Conjugated enynes as nonaromat ...... referentially the D(3) subtype
@en
Conjugated enynes as nonaromat ...... referentially the D(3) subtype
@nl
P2093
P3181
P356
P1476
Conjugated enynes as nonaromat ...... referentially the D(3) subtype
@en
P2093
P304
P3181
P356
10.1021/JM991098Z
P407
P577
2000-02-24T00:00:00Z