Structural basis of N-Myc binding by Aurora-A and its destabilization by kinase inhibitors.
about
Time, space, and disorder in the expanding proteome universe.MYC Deregulation in Primary Human Cancers.Neuroblastoma treatment in the post-genomic era.Drugging the 'undruggable' cancer targets.Cisplatin-resistant cancer cells are sensitive to Aurora kinase A inhibition by alisertib.The importance of regulatory ubiquitination in cancer and metastasis.Switching Aurora-A kinase on and off at an allosteric site.The MYCN Protein in Health and Disease.Dynamic Equilibrium of the Aurora A Kinase Activation Loop Revealed by Single-Molecule Spectroscopy.Integrated Molecular Meta-Analysis of 1,000 Pediatric High-Grade and Diffuse Intrinsic Pontine Glioma.Association with Aurora-A Controls N-MYC-Dependent Promoter Escape and Pause Release of RNA Polymerase II during the Cell Cycle.Multivariate analysis of risk factors for patients with stage 4 neuroblastoma who were older than 18 months at diagnosis: a report from a single institute in Shanghai, China.A dynamic mechanism for allosteric activation of Aurora kinase A by activation loop phosphorylation.Mitotic spindle association of TACC3 requires Aurora-A-dependent stabilization of a cryptic α-helix.The multifaceted allosteric regulation of Aurora kinase A.
P2860
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P2860
Structural basis of N-Myc binding by Aurora-A and its destabilization by kinase inhibitors.
description
2016 nî lūn-bûn
@nan
2016 թուականի Նոյեմբերին հրատարակուած գիտական յօդուած
@hyw
2016 թվականի նոյեմբերին հրատարակված գիտական հոդված
@hy
2016年の論文
@ja
2016年論文
@yue
2016年論文
@zh-hant
2016年論文
@zh-hk
2016年論文
@zh-mo
2016年論文
@zh-tw
2016年论文
@wuu
name
Structural basis of N-Myc bind ...... lization by kinase inhibitors.
@ast
Structural basis of N-Myc bind ...... lization by kinase inhibitors.
@en
Structural basis of N-Myc bind ...... lization by kinase inhibitors.
@en-gb
type
label
Structural basis of N-Myc bind ...... lization by kinase inhibitors.
@ast
Structural basis of N-Myc bind ...... lization by kinase inhibitors.
@en
Structural basis of N-Myc bind ...... lization by kinase inhibitors.
@en-gb
prefLabel
Structural basis of N-Myc bind ...... lization by kinase inhibitors.
@ast
Structural basis of N-Myc bind ...... lization by kinase inhibitors.
@en
Structural basis of N-Myc bind ...... lization by kinase inhibitors.
@en-gb
P2860
P50
P356
P1154
2-s2.0-84999188126
P1476
Structural basis of N-Myc bind ...... lization by kinase inhibitors.
@en
P2093
Anne Carstensen
Martin Eilers
P2860
P304
13726-13731
P356
10.1073/PNAS.1610626113
P407
P5530
P577
2016-11-11T00:00:00Z
P6179
1002230036