Small molecule biaryl FSH receptor agonists. Part 1: Lead discovery via encoded combinatorial synthesis.
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Discovery and Development of Small Molecule Allosteric Modulators of Glycoprotein Hormone ReceptorsAllosteric activation of the follicle-stimulating hormone (FSH) receptor by selective, nonpeptide agonists.Human TSH receptor ligands as pharmacological probes with potential clinical applicationA negative allosteric modulator demonstrates biased antagonism of the follicle stimulating hormone receptor.Solid-phase and microwave-assisted syntheses of 2,5-diketopiperazines: small molecules with great potentialSmall-molecule agonists for the thyrotropin receptor stimulate thyroid function in human thyrocytes and mice.Novel pathways in gonadotropin receptor signaling and biased agonism.Development of Selective LH Receptor Agonists by Heterodimerization with a FSH Receptor Antagonist.Induction of ovulation by a potent, orally active, low molecular weight agonist (Org 43553) of the luteinizing hormone receptor.Synthesis and pharmacological evaluation of dimeric follicle-stimulating hormone receptor antagonists.
P2860
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P2860
Small molecule biaryl FSH receptor agonists. Part 1: Lead discovery via encoded combinatorial synthesis.
description
2004 nî lūn-bûn
@nan
2004 թուականի Ապրիլին հրատարակուած գիտական յօդուած
@hyw
2004 թվականի ապրիլին հրատարակված գիտական հոդված
@hy
2004年の論文
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2004年論文
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2004年論文
@zh-hant
2004年論文
@zh-hk
2004年論文
@zh-mo
2004年論文
@zh-tw
2004年论文
@wuu
name
Small molecule biaryl FSH rece ...... coded combinatorial synthesis.
@ast
Small molecule biaryl FSH rece ...... coded combinatorial synthesis.
@en
type
label
Small molecule biaryl FSH rece ...... coded combinatorial synthesis.
@ast
Small molecule biaryl FSH rece ...... coded combinatorial synthesis.
@en
prefLabel
Small molecule biaryl FSH rece ...... coded combinatorial synthesis.
@ast
Small molecule biaryl FSH rece ...... coded combinatorial synthesis.
@en
P2093
P1476
Small molecule biaryl FSH rece ...... coded combinatorial synthesis.
@en
P2093
Anton E P Adang
Brian F McGuinness
Dan Fitzpatrick
Edward McDonald
Guizhen Dong
Kenneth J Valenzano
Koc-Kan Ho
Kurt W Saionz
Maria L Webb
P304
P356
10.1016/J.BMCL.2004.01.042
P407
P577
2004-04-01T00:00:00Z