Identification of a peptoid inhibitor of the proteasome 19S regulatory particle.
about
Variably modulated gating of the 26S proteasome by ATP and polyubiquitinTowards vast libraries of scaffold-diverse, conformationally constrained oligomers.High-throughput evaluation of relative cell permeability between peptoids and peptides.Encoded combinatorial libraries for the construction of cyclic peptoid microarraysDiscovering ligands for a microRNA precursor with peptoid microarrays.Utility of redundant combinatorial libraries in distinguishing high and low quality screening hitsPeptoid ligands that bind selectively to phosphoproteins.Development of homomultimers and heteromultimers of lung cancer-specific peptoids.On-Bead Two-Color (OBTC) Cell Screen for Direct Identification of Highly Selective Cell Surface Receptor Ligands.Synthesis of libraries of peptidomimetic compounds containing a 2-oxopiperazine unit in the main chain.On-bead screens sample narrower affinity ranges of protein-ligand interactions compared to equivalent solution assays.Aβ42-binding peptoids as amyloid aggregation inhibitors and detection ligands.Potent and selective photo-inactivation of proteins with peptoid-ruthenium conjugates.Discovery of peptoid ligands for anti-aquaporin 4 antibodiesSynthesis and screening of stereochemically diverse combinatorial libraries of peptide tertiary amides.Proteome dynamics and proteome function of cardiac 19S proteasomesInfluencing uptake and localization of aminoglycoside-functionalized peptoids.The identification of high-affinity G protein-coupled receptor ligands from large combinatorial libraries using multicolor quantum dot-labeled cell-based screening.Split-and-pool synthesis and characterization of peptide tertiary amide libraryExpanded polyglutamine-binding peptoid as a novel therapeutic agent for treatment of Huntington's disease.Positional Scanning Synthesis of a Peptoid Library Yields New Inducers of Apoptosis that Target Karyopherins and Tubulin.In-Bead Screening of Hydroxamic Acids for the Identification of HDAC Inhibitors.Development of a large peptoid-DOTA combinatorial library.Discovery of an Inhibitor of the Proteasome Subunit Rpn11.Periodate-triggered cross-linking reveals Sug2/Rpt4 as the molecular target of a peptoid inhibitor of the 19S proteasome regulatory particle.Sophistication of foldamer form and function in vitro and in vivo.Structure-function relationships in peptoids: recent advances toward deciphering the structural requirements for biological function.Non-proteolytic regulation of p53-mediated transcription through destabilization of the activator.promoter complex by the proteasomal ATPases.Synthetic receptors with antibody-like binding affinities.Heterogeneous cardiac proteasomes: mandated by diverse substrates?Peptides and proteins as a continuing exciting source of inspiration for peptidomimetics.Peptide and peptoid foldamers in medicinal chemistry.Establishment of a suite of assays that support the discovery of proteasome stimulators.A reversible and highly selective inhibitor of the proteasomal ubiquitin receptor rpn13 is toxic to multiple myeloma cellsAn overview of peptide and peptoid foldamers in medicinal chemistry.Extraordinarily robust polyproline type I peptoid helices generated via the incorporation of α-chiral aromatic N-1-naphthylethyl side chains.Selective anticancer copper(II)-mixed ligand complexes: targeting of ROS and proteasomes.Design and conformational analysis of peptoids containing N-hydroxy amides reveals a unique sheet-like secondary structure.Capzimin is a potent and specific inhibitor of proteasome isopeptidase Rpn11.A general system for evaluating the efficiency of chromophore-assisted light inactivation (CALI) of proteins reveals Ru(II) tris-bipyridyl as an unusually efficient "warhead".
P2860
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P2860
Identification of a peptoid inhibitor of the proteasome 19S regulatory particle.
description
2007 nî lūn-bûn
@nan
2007 թուականի Մայիսին հրատարակուած գիտական յօդուած
@hyw
2007 թվականի մայիսին հրատարակված գիտական հոդված
@hy
2007年の論文
@ja
2007年論文
@yue
2007年論文
@zh-hant
2007年論文
@zh-hk
2007年論文
@zh-mo
2007年論文
@zh-tw
2007年论文
@wuu
name
Identification of a peptoid inhibitor of the proteasome 19S regulatory particle.
@ast
Identification of a peptoid inhibitor of the proteasome 19S regulatory particle.
@en
type
label
Identification of a peptoid inhibitor of the proteasome 19S regulatory particle.
@ast
Identification of a peptoid inhibitor of the proteasome 19S regulatory particle.
@en
prefLabel
Identification of a peptoid inhibitor of the proteasome 19S regulatory particle.
@ast
Identification of a peptoid inhibitor of the proteasome 19S regulatory particle.
@en
P2093
P2860
P356
P1476
Identification of a peptoid inhibitor of the proteasome 19S regulatory particle.
@en
P2093
Chase T Archer
Hyun-Suk Lim
Thomas Kodadek
P2860
P304
P356
10.1021/JA072027P
P407
P577
2007-05-31T00:00:00Z