Discovery of N-{[1-(propylsulfonyl)-4-pyridin-2-ylpiperidin-4-yl]methyl}benzamides as novel, selective and potent GlyT1 inhibitors.
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Novel GlyT1 inhibitor chemotypes by scaffold hopping. Part 1: development of a potent and CNS penetrant [3.1.0]-based lead.Glutamatergic targets for enhancing extinction learning in drug addictionNovel GlyT1 inhibitor chemotypes by scaffold hopping. Part 2: development of a [3.3.0]-based series and other piperidine bioisosteresThe synthesis and preclinical evaluation in rhesus monkey of [¹⁸F]MK-6577 and [¹¹C]CMPyPB glycine transporter 1 positron emission tomography radiotracers.Copper-Catalyzed Alkylation of Nitroalkanes with α-Bromonitriles: Synthesis of β-Cyanonitroalkanes.Metabolism-guided drug design
P2860
Discovery of N-{[1-(propylsulfonyl)-4-pyridin-2-ylpiperidin-4-yl]methyl}benzamides as novel, selective and potent GlyT1 inhibitors.
description
2009 nî lūn-bûn
@nan
2009 թուականի Յունուարին հրատարակուած գիտական յօդուած
@hyw
2009 թվականի հունվարին հրատարակված գիտական հոդված
@hy
2009年の論文
@ja
2009年論文
@yue
2009年論文
@zh-hant
2009年論文
@zh-hk
2009年論文
@zh-mo
2009年論文
@zh-tw
2009年论文
@wuu
name
Discovery of N-{[1-(propylsulf ...... e and potent GlyT1 inhibitors.
@ast
Discovery of N-{[1-(propylsulf ...... e and potent GlyT1 inhibitors.
@en
type
label
Discovery of N-{[1-(propylsulf ...... e and potent GlyT1 inhibitors.
@ast
Discovery of N-{[1-(propylsulf ...... e and potent GlyT1 inhibitors.
@en
prefLabel
Discovery of N-{[1-(propylsulf ...... e and potent GlyT1 inhibitors.
@ast
Discovery of N-{[1-(propylsulf ...... e and potent GlyT1 inhibitors.
@en
P2093
P1476
Discovery of N-{[1-(propylsulf ...... e and potent GlyT1 inhibitors.
@en
P2093
Cyrille Sur
David L Williams
Doug J Pettibone
Gene G Kinney
George D Hartman
Julie A O'Brien
Marlene A Jacobson
Philip R Tiller
Scott E Wolkenberg
Sheri Smith
P304
P356
10.1016/J.BMCL.2008.12.115
P407
P577
2009-01-09T00:00:00Z