Pungency of TRPV1 agonists is directly correlated with kinetics of receptor activation and lipophilicity.
about
TRPV1: A Target for Rational Drug DesignThe involvement of TRPV1 in emesis and anti-emesisCannabinoid-based drugs targeting CB1 and TRPV1, the sympathetic nervous system, and arthritisEffects of cannabinoids and cannabinoid-enriched Cannabis extracts on TRP channels and endocannabinoid metabolic enzymes.Capsaicin interaction with TRPV1 channels in a lipid bilayer: molecular dynamics simulation.Chemosensory properties of the trigeminal system.N-glycosylation determines ionic permeability and desensitization of the TRPV1 capsaicin receptor.Thermosensitive transient receptor potential (TRP) channel agonists and their role in mechanical, thermal and nociceptive sensations as assessed using animal models.Anti-nociceptive and desensitizing effects of olvanil on capsaicin-induced thermal hyperalgesia in the rat.The Alkamide trans-Pellitorine Targets PPARγ via TRPV1 and TRPA1 to Reduce Lipid Accumulation in Developing 3T3-L1 Adipocytes.Structure-Driven Pharmacology of Transient Receptor Potential Channel Vanilloid 1.Tasty and healthy TR(i)Ps. The human quest for culinary pungency.Effect of chirality and lipophilicity in the functional activity of evodiamine and its analogues at TRPV1 channels.Primary alcohols activate human TRPA1 channel in a carbon chain length-dependent manner.Photoswitchable fatty acids enable optical control of TRPV1.Characterisation of Nav1.7 functional expression in rat dorsal root ganglia neurons by using an electrical field stimulation assay.TRPA1-dependent reversible opening of tight junction by natural compounds with an α,β-unsaturated moiety and capsaicin.Isolation and identification of a humanTRPV1 activating compound from soy sauce.Naturally Produced Defensive Alkenal Compounds Activate TRPA1.Utility of in vitro and in vivo systems for studying the permeability of capsaicin and nonivamide through different intestinal regions.Pharmacodynamics of TRPV1 agonists in a bioassay using human PC-3 cells.Chemical Activation of Sensory TRP Channels
P2860
Q26738621-A2E1D65F-01D9-4ACC-9806-48B4692566E5Q26745801-C0AAA802-35AF-4A29-961A-FAE747F477B1Q26783956-89010800-D843-4315-BC58-D6AAFA974348Q34625932-933969F4-7DDF-45D7-BDC4-0A9A239109FBQ35221694-8621539B-0736-4B9C-95F5-51F02278BF39Q36015318-C286ABFE-CA5A-412F-9F93-6F422B0EACA1Q36052386-802976BA-EA43-42C0-A735-8B6AB24F5D7FQ36067431-6A3D2BB5-892F-4DC0-8B4D-F1442F2E64CCQ36083250-FE7A27F3-3178-4142-9898-1E32379538AEQ38723177-B86266F7-4032-4234-B8EF-51CBAF891F69Q38874068-DB601C77-3C0B-4B92-A331-CB27F633ED6EQ38922657-A88EE3BD-8499-46EE-BB03-3DFE5ADDED09Q39189093-87D78A4F-DC94-4D8A-96E9-C8BD4CB5F3D5Q39416776-82DED5F1-D764-455E-9316-36A1079527A7Q42089811-FABC386E-B01E-406B-B9BB-C0D779109F04Q47113350-96BC0B7D-14C3-477F-8B9C-498F8A1E06B4Q49357566-A6DBFE76-12CC-4CCE-A6AE-5F42238E0715Q50218822-0FC496B5-815D-4CDC-B02B-20660BE50A1FQ50536040-6994863F-09E1-4AC5-8C3E-632E49819EAFQ50579051-C44E21E3-9A50-46F8-90E3-C3038A38DD62Q51098262-89A650BE-728C-4BF7-A252-52DA3E4B0F50Q56552616-3490AFA9-8CC4-410A-BF26-D163FA87248D
P2860
Pungency of TRPV1 agonists is directly correlated with kinetics of receptor activation and lipophilicity.
description
2010 nî lūn-bûn
@nan
2010 թուականի Յունիսին հրատարակուած գիտական յօդուած
@hyw
2010 թվականի հունիսին հրատարակված գիտական հոդված
@hy
2010年の論文
@ja
2010年論文
@yue
2010年論文
@zh-hant
2010年論文
@zh-hk
2010年論文
@zh-mo
2010年論文
@zh-tw
2010年论文
@wuu
name
Pungency of TRPV1 agonists is ...... activation and lipophilicity.
@ast
Pungency of TRPV1 agonists is ...... activation and lipophilicity.
@en
type
label
Pungency of TRPV1 agonists is ...... activation and lipophilicity.
@ast
Pungency of TRPV1 agonists is ...... activation and lipophilicity.
@en
prefLabel
Pungency of TRPV1 agonists is ...... activation and lipophilicity.
@ast
Pungency of TRPV1 agonists is ...... activation and lipophilicity.
@en
P2093
P1476
Pungency of TRPV1 agonists is ...... activation and lipophilicity.
@en
P2093
Daniel Ursu
Emanuele Sher
Kelly Knopp
Ruth E Beattie
P304
P356
10.1016/J.EJPHAR.2010.05.029
P407
P577
2010-06-08T00:00:00Z