Monepantel allosterically activates DEG-3/DES-2 channels of the gastrointestinal nematode Haemonchus contortus.
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Principles of agonist recognition in Cys-loop receptorsPhylogenomics of ligand-gated ion channels predicts monepantel effectFunctional Characterization of a Novel Class of Morantel-Sensitive Acetylcholine Receptors in NematodesCuriouser and Curiouser: The Macrocyclic Lactone, Abamectin, Is also a Potent Inhibitor of Pyrantel/Tribendimidine Nicotinic Acetylcholine Receptors of Gastro-Intestinal Wormsacr-23 Encodes a monepantel-sensitive channel in Caenorhabditis elegans.The Ascaris suum nicotinic receptor, ACR-16, as a drug target: Four novel negative allosteric modulators from virtual screening.Ion channels and receptor as targets for the control of parasitic nematodes.Betaine acts on a ligand-gated ion channel in the nervous system of the nematode C. elegans.Neurobiology of plant parasitic nematodes.Discovery and development of veterinary antiparasitic drugs: past, present and future.The evolution of pentameric ligand-gated ion-channels and the changing family of anthelmintic drug targets.Acquired resistance to monepantel in C. elegans: What about parasitic nematodes?Anticancer properties of novel aminoacetonitrile derivative monepantel (ADD 1566) in pre-clinical models of human ovarian cancer.Monepantel induces autophagy in human ovarian cancer cells through disruption of the mTOR/p70S6K signalling pathwayMonepantel is a non-competitive antagonist of nicotinic acetylcholine receptors from Ascaris suum and Oesophagostomum dentatum.A BRIEF REVIEW ON THE MODE OF ACTION OF ANTINEMATODAL DRUGS.
P2860
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P2860
Monepantel allosterically activates DEG-3/DES-2 channels of the gastrointestinal nematode Haemonchus contortus.
description
2010 nî lūn-bûn
@nan
2010 թուականի Օգոստոսին հրատարակուած գիտական յօդուած
@hyw
2010 թվականի օգոստոսին հրատարակված գիտական հոդված
@hy
2010年の論文
@ja
2010年論文
@yue
2010年論文
@zh-hant
2010年論文
@zh-hk
2010年論文
@zh-mo
2010年論文
@zh-tw
2010年论文
@wuu
name
Monepantel allosterically acti ...... nematode Haemonchus contortus.
@ast
Monepantel allosterically acti ...... nematode Haemonchus contortus.
@en
type
label
Monepantel allosterically acti ...... nematode Haemonchus contortus.
@ast
Monepantel allosterically acti ...... nematode Haemonchus contortus.
@en
prefLabel
Monepantel allosterically acti ...... nematode Haemonchus contortus.
@ast
Monepantel allosterically acti ...... nematode Haemonchus contortus.
@en
P2093
P356
P1476
Monepantel allosterically acti ...... nematode Haemonchus contortus.
@en
P2093
Erwin Sigel
Lucien Rufener
Roland Baur
Ronald Kaminsky
P304
P356
10.1124/MOL.110.066498
P50
P577
2010-08-02T00:00:00Z