Pasireotide and octreotide stimulate distinct patterns of sst2A somatostatin receptor phosphorylation.
about
The effects of somatostatin analogue therapy on pituitary tumor volume in patients with acromegalyPI3K-AKT-mTOR-signaling and beyond: the complex network in gastroenteropancreatic neuroendocrine neoplasmsNanoparticle ligand presentation for targeting solid tumorsFine-tuning somatostatin receptor signalling by agonist-selective phosphorylation and dephosphorylation: IUPHAR Review 5Somatostatin Depresses the Excitability of Subicular Bursting Cells: Roles of Inward Rectifier K+ Channels, KCNQ channels and Epac.A transplantable phosphorylation probe for direct assessment of G protein-coupled receptor activation.Hierarchical organization of multi-site phosphorylation at the CXCR4 C terminus.Ligand-dependent mechanisms of sst2A receptor trafficking: role of site-specific phosphorylation and receptor activation in the actions of biased somatostatin agonists.Phase II study of monthly pasireotide LAR (SOM230C) for recurrent or progressive meningioma.Differentiation of opioid drug effects by hierarchical multi-site phosphorylationIlluminating somatostatin analog action at neuroendocrine tumor receptorsHeterologous regulation of agonist-independent μ-opioid receptor phosphorylation by protein kinase CPasireotide for the treatment of Cushing's disease.Somatostatin receptor biology in neuroendocrine and pituitary tumours: part 2--clinical implicationsDetermination of GPCR Phosphorylation Status: Establishing a Phosphorylation Barcode.Rapid dephosphorylation of G protein-coupled receptors by protein phosphatase 1β is required for termination of β-arrestin-dependent signaling.Identification of human somatostatin receptor 2 domains involved in internalization and signaling in QGP-1 pancreatic neuroendocrine tumor cell line.Inhibition of Peripheral Synthesis of Serotonin as a New Target in Neuroendocrine Tumors.Pasireotide is more effective than octreotide, alone or combined with everolimus on human meningioma in vitroDeciphering µ-opioid receptor phosphorylation and dephosphorylation in HEK293 cells.Structural determinants of agonist-selective signaling at the sst(2A) somatostatin receptor.Phosphorylation of threonine 333 regulates trafficking of the human sst5 somatostatin receptorIdentification of Phosphorylation Sites Regulating sst3 Somatostatin Receptor Trafficking.Differential regulation of somatostatin receptor dephosphorylation by β-arrestin1 and β-arrestin2.Reassessment of sst3 somatostatin receptor expression in human normal and neoplastic tissues using the novel rabbit monoclonal antibody UMB-5.Effects of pasireotide (SOM230) on protein turnover and p70S6 kinase-S6 ribosomal protein signaling pathway in rat skeletal muscle cells.International Union of Basic and Clinical Pharmacology. CV. Somatostatin Receptors: Structure, Function, Ligands, and New Nomenclature
P2860
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P2860
Pasireotide and octreotide stimulate distinct patterns of sst2A somatostatin receptor phosphorylation.
description
2010 nî lūn-bûn
@nan
2010 թուականի Յունուարին հրատարակուած գիտական յօդուած
@hyw
2010 թվականի հունվարին հրատարակված գիտական հոդված
@hy
2010年の論文
@ja
2010年論文
@yue
2010年論文
@zh-hant
2010年論文
@zh-hk
2010年論文
@zh-mo
2010年論文
@zh-tw
2010年论文
@wuu
name
Pasireotide and octreotide sti ...... atin receptor phosphorylation.
@ast
Pasireotide and octreotide sti ...... atin receptor phosphorylation.
@en
type
label
Pasireotide and octreotide sti ...... atin receptor phosphorylation.
@ast
Pasireotide and octreotide sti ...... atin receptor phosphorylation.
@en
prefLabel
Pasireotide and octreotide sti ...... atin receptor phosphorylation.
@ast
Pasireotide and octreotide sti ...... atin receptor phosphorylation.
@en
P2093
P2860
P356
P1476
Pasireotide and octreotide sti ...... atin receptor phosphorylation.
@en
P2093
Amelie Lupp
Diana Lehmann
Florian Pöll
Mihaela Ginj
Ralf Stumm
Stefan Jacobs
Stefan Schulz
Susann Illing
P2860
P304
P356
10.1210/ME.2009-0315
P577
2010-01-05T00:00:00Z