Desensitization of functional µ-opioid receptors increases agonist off-rate.
about
Opioid receptor desensitization: mechanisms and its link to toleranceAgonist Binding and Desensitization of the μ-Opioid Receptor Is Modulated by Phosphorylation of the C-Terminal Tail Domain.Differential desensitization observed at multiple effectors of somatic mu opioid receptors underlies sustained agonist-mediated inhibition of proopiomelanocortin neuron activity.New Technologies for Elucidating Opioid Receptor Function.Desensitization and tolerance of mu opioid receptors on pontine Kolliker-Fuse neurons.A Caged Enkephalin Optimized for Simultaneously Probing Mu and Delta Opioid Receptors.Cellular tolerance at the µ-opioid receptor is phosphorylation dependent.
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Q34729984-D24DB45C-AC94-48B8-8937-CC3FDA9C6C46Q36077748-DB7ABBE6-16FD-4FA9-9C7C-CD81EDF26E9AQ38617993-041835EA-F65A-4CDD-B35D-D17ED22981E2Q38718788-8F17AB92-9025-478A-9AC2-84B286DF1688Q44350406-DDEF035C-272A-47DE-BE67-3762A8F0D6B0Q47902030-9F5A7ABB-0A9A-4F79-A662-0C41A7D6C740Q54246867-9DC558D8-0B2C-4D6E-8ABE-8790A66D3E89
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Desensitization of functional µ-opioid receptors increases agonist off-rate.
description
2014 nî lūn-bûn
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2014 թուականի Ապրիլին հրատարակուած գիտական յօդուած
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2014 թվականի ապրիլին հրատարակված գիտական հոդված
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2014年の論文
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2014年論文
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2014年論文
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2014年論文
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2014年論文
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2014年論文
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2014年论文
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name
Desensitization of functional µ-opioid receptors increases agonist off-rate.
@ast
Desensitization of functional µ-opioid receptors increases agonist off-rate.
@en
type
label
Desensitization of functional µ-opioid receptors increases agonist off-rate.
@ast
Desensitization of functional µ-opioid receptors increases agonist off-rate.
@en
prefLabel
Desensitization of functional µ-opioid receptors increases agonist off-rate.
@ast
Desensitization of functional µ-opioid receptors increases agonist off-rate.
@en
P2860
P356
P1476
Desensitization of functional µ-opioid receptors increases agonist off-rate.
@en
P2093
John T Williams
P2860
P356
10.1124/MOL.114.092098
P577
2014-04-18T00:00:00Z