Overlap between the ligand recognition properties of the anandamide transporter and the VR1 vanilloid receptor: inhibitors of anandamide uptake with negligible capsaicin-like activity.
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An endogenous capsaicin-like substance with high potency at recombinant and native vanilloid VR1 receptors.Novel bioactive metabolites of dipyrone (metamizol)The endocannabinoid system as a target for the treatment of cannabis dependenceThe endocannabinoid system as an emerging target of pharmacotherapyAM404, an inhibitor of anandamide uptake, prevents pain behaviour and modulates cytokine and apoptotic pathways in a rat model of neuropathic painEvidence against the presence of an anandamide transporterFunctionally important amino acid residues in the transient receptor potential vanilloid 1 (TRPV1) ion channel--an overview of the current mutational data"Redundancy" of endocannabinoid inactivation: new challenges and opportunities for pain controlTRPV1 in brain is involved in acetaminophen-induced antinociceptionConversion of acetaminophen to the bioactive N-acylphenolamine AM404 via fatty acid amide hydrolase-dependent arachidonic acid conjugation in the nervous systemThe endocannabinoid/endovanilloid N-arachidonoyl dopamine (NADA) and synthetic cannabinoid WIN55,212-2 abate the inflammatory activation of human endothelial cellsInternational Union of Basic and Clinical Pharmacology. LXXIX. Cannabinoid receptors and their ligands: beyond CB₁ and CB₂Palmitoylethanolamide inhibits the expression of fatty acid amide hydrolase and enhances the anti-proliferative effect of anandamide in human breast cancer cellsEffects of homologues and analogues of palmitoylethanolamide upon the inactivation of the endocannabinoid anandamideMolecular targets for cannabidiol and its synthetic analogues: effect on vanilloid VR1 receptors and on the cellular uptake and enzymatic hydrolysis of anandamideCharacterization of palmitoylethanolamide transport in mouse Neuro-2a neuroblastoma and rat RBL-2H3 basophilic leukaemia cells: comparison with anandamideFatty acid amide hydrolase-dependent generation of antinociceptive drug metabolites acting on TRPV1 in the brainRequirement for the endocannabinoid system in social interaction impairment induced by coactivation of dopamine D1 and D2 receptors in the piriform cortexRole of Cannabinoids in Gastrointestinal Mucosal Defense and InflammationEndocannabinoid signalling in reward and addiction.Differential effect of cannabinoid agonists and endocannabinoids on histamine release from distinct regions of the rat brainInhibition of human recombinant T-type calcium channels by the endocannabinoid N-arachidonoyl dopamine.AM404 attenuates reinstatement of nicotine seeking induced by nicotine-associated cues and nicotine priming but does not affect nicotine- and food-taking.Anandamide acts as an intracellular messenger amplifying Ca2+ influx via TRPV1 channels.Binding, degradation and apoptotic activity of stearoylethanolamide in rat C6 glioma cells.The endogenous cannabinoid, anandamide, inhibits dopamine transporter function by a receptor-independent mechanism.N-arachidonyl-glycine modulates synaptic transmission in superficial dorsal hornEndocannabinoid-dependent LTD in a nociceptive synapse requires activation of a presynaptic TRPV-like receptor.Cannabinoid receptors as target for treatment of osteoporosis: a tale of two therapies.An endocannabinoid mechanism for stress-induced analgesia.Anandamide uptake is consistent with rate-limited diffusion and is regulated by the degree of its hydrolysis by fatty acid amide hydrolase.Acetaminophen from liver to brain: New insights into drug pharmacological action and toxicityRole of endocannabinoids and cannabinoid-1 receptors in cerebrocortical blood flow regulation.Vascular effects of anandamide and N-acylvanillylamines in the human forearm and skin microcirculation.Acetaminophen modulation of hydrocodone reward in rats.New potent and selective inhibitors of anandamide reuptake with antispastic activity in a mouse model of multiple sclerosisCannabinoids and cancer: pros and cons of an antitumour strategy.Identification of a binding motif in the S5 helix that confers cholesterol sensitivity to the TRPV1 ion channel.Cellular accumulation of anandamide: consensus and controversy.The selective anandamide transport inhibitor VDM11 attenuates reinstatement of nicotine seeking behaviour, but does not affect nicotine intake
P2860
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P2860
Overlap between the ligand recognition properties of the anandamide transporter and the VR1 vanilloid receptor: inhibitors of anandamide uptake with negligible capsaicin-like activity.
description
2000 nî lūn-bûn
@nan
2000 թուականի Հոկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2000 թվականի հոտեմբերին հրատարակված գիտական հոդված
@hy
2000年の論文
@ja
2000年論文
@yue
2000年論文
@zh-hant
2000年論文
@zh-hk
2000年論文
@zh-mo
2000年論文
@zh-tw
2000年论文
@wuu
name
Overlap between the ligand rec ...... gible capsaicin-like activity.
@ast
Overlap between the ligand rec ...... gible capsaicin-like activity.
@en
type
label
Overlap between the ligand rec ...... gible capsaicin-like activity.
@ast
Overlap between the ligand rec ...... gible capsaicin-like activity.
@en
prefLabel
Overlap between the ligand rec ...... gible capsaicin-like activity.
@ast
Overlap between the ligand rec ...... gible capsaicin-like activity.
@en
P2093
P2860
P1433
P1476
Overlap between the ligand rec ...... gible capsaicin-like activity.
@en
P2093
L De Petrocellis
R G Pertwee
V Di Marzo
P2860
P356
10.1016/S0014-5793(00)02082-2
P407
P577
2000-10-01T00:00:00Z