High constitutive activity of native H3 receptors regulates histamine neurons in brain.
about
Loss of constitutive activity of the growth hormone secretagogue receptor in familial short statureG protein-coupled receptors in the hypothalamic paraventricular and supraoptic nuclei--serpentine gateways to neuroendocrine homeostasisThe histamine H3 receptor: an attractive target for the treatment of cognitive disordersHistamine and its receptorsAcute wake-promoting actions of JNJ-5207852, a novel, diamine-based H3 antagonistDetection of multiple H3 receptor affinity states utilizing [3H]A-349821, a novel, selective, non-imidazole histamine H3 receptor inverse agonist radioligandPlasticity of histamine H3 receptor expression and binding in the vestibular nuclei after labyrinthectomy in ratIncreased brain histamine H3 receptor expression during hibernation in golden-mantled ground squirrelsEnhanced spontaneous activity of the mu opioid receptor by cysteine mutations: characterization of a tool for inverse agonist screeningHistaminergic mechanisms for modulation of memory systemsPhasic and Tonic mGlu7 Receptor Activity Modulates the Thalamocortical NetworkThe Subcellular Dynamics of the Gs-Linked Receptor GPR3 Contribute to the Local Activation of PKA in Cerebellar Granular NeuronsTwo polymorphic forms of human histamine methyltransferase: structural, thermal, and kinetic comparisonsMonoaminergic and Histaminergic Strategies and Treatments in Brain DiseasesThe cell biology of acute itchConstitutive activation of A(3) adenosine receptors by site-directed mutagenesisThe role of carcinine in signaling at the Drosophila photoreceptor synapseInteractions between histamine H3 and dopamine D2 receptors and the implications for striatal functionGenetic Analysis of Histamine Signaling in Larval Zebrafish Sleep.Identification of inhibitors of Plasmodium falciparum phosphoethanolamine methyltransferase using an enzyme-coupled transmethylation assay.The histaminergic system is involved in psychological stress-induced hyperthermia in rats.Structural basis for inhibition of histamine N-methyltransferase by diverse drugsCannabinoid CB1 receptor-interacting proteins: novel targets for central nervous system drug discovery?H1-antihistamines: inverse agonism, anti-inflammatory actions and cardiac effects.Histamine in the regulation of wakefulness.BML-190 and AM251 act as inverse agonists at the human cannabinoid CB2 receptor: signalling via cAMP and inositol phosphates.Inverse agonism and its therapeutic significance.Protean agonism at histamine H3 receptors in vitro and in vivoThe rat cytomegalovirus R33-encoded G protein-coupled receptor signals in a constitutive fashionPerspectives on cognitive domains, H3 receptor ligands and neurological disease.The histamine H3 receptor: from gene cloning to H3 receptor drugs.H3 receptors and pain modulation: peripheral, spinal, and brain interactions.Genetic variations in human G protein-coupled receptors: implications for drug therapy.Altered sleep-wake characteristics and lack of arousal response to H3 receptor antagonist in histamine H1 receptor knockout mice.Dimer-dependent intrinsic/basal activity of the class B G protein-coupled receptor PAC1 promotes cellular anti-apoptotic activity through Wnt/β-catenin pathways that are associated with dimer endocytosisThe histamine H3 receptor: from discovery to clinical trials with pitolisantHomer as both a scaffold and transduction molecule.LC-MS/MS method for the determination of pitolisant: application to rat pharmacokinetic and brain penetration studies.G-protein-coupled receptors: past, present and future.Inverse agonists: tools to reveal ligand-specific conformations of G protein-coupled receptors.
P2860
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P2860
High constitutive activity of native H3 receptors regulates histamine neurons in brain.
description
2000 nî lūn-bûn
@nan
2000 թուականի Դեկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2000 թվականի դեկտեմբերին հրատարակված գիտական հոդված
@hy
2000年の論文
@ja
2000年論文
@yue
2000年論文
@zh-hant
2000年論文
@zh-hk
2000年論文
@zh-mo
2000年論文
@zh-tw
2000年论文
@wuu
name
High constitutive activity of native H3 receptors regulates histamine neurons in brain.
@ast
High constitutive activity of native H3 receptors regulates histamine neurons in brain.
@en
type
label
High constitutive activity of native H3 receptors regulates histamine neurons in brain.
@ast
High constitutive activity of native H3 receptors regulates histamine neurons in brain.
@en
prefLabel
High constitutive activity of native H3 receptors regulates histamine neurons in brain.
@ast
High constitutive activity of native H3 receptors regulates histamine neurons in brain.
@en
P2093
P2860
P356
P1433
P1476
High constitutive activity of native H3 receptors regulates histamine neurons in brain
@en
P2093
Ganellin CR
Morisset S
Schunack W
Schwartz JC
Tardivel-Lacombe J
P2860
P2888
P304
P356
10.1038/35048583
P407
P577
2000-12-01T00:00:00Z
P5875
P6179
1020002135