International Union of Basic and Clinical Pharmacology. LXXXII: Nomenclature and Classification of Hydroxy-carboxylic Acid Receptors (GPR81, GPR109A, and GPR109B).
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International Union of Basic and Clinical Pharmacology. LXXXVIII. G protein-coupled receptor list: recommendations for new pairings with cognate ligandsRole of β-hydroxybutyrate, its polymer poly-β-hydroxybutyrate and inorganic polyphosphate in mammalian health and diseaseLactate transport and signaling in the brain: potential therapeutic targets and roles in body-brain interactionGPR109A and vascular inflammationThe eosinophil chemoattractant 5-oxo-ETE and the OXE receptorNaturally occurring HCA1 missense mutations result in loss of function: potential impact on lipid deposition.The Concise Guide to PHARMACOLOGY 2013/14: G protein-coupled receptorsKetone bodies as signaling metabolites.Redistribution of monocarboxylate transporter 2 on the surface of astrocytes in the human epileptogenic hippocampusHydroxycarboxylic acid receptor 2 mediates dimethyl fumarate's protective effect in EAE.Nicotinic acid receptor GPR109A is down-regulated in human macrophage-derived foam cells.β-hydroxybutyrate: much more than a metaboliteIFNγ Induces DNA Methylation-Silenced GPR109A Expression via pSTAT1/p300 and H3K18 Acetylation in Colon Cancer.Biological roles and therapeutic potential of hydroxy-carboxylic Acid receptors.Niacin in cardiovascular disease: recent preclinical and clinical developmentsPlasma Metabolites Predict Severity of Depression and Suicidal Ideation in Psychiatric Patients-A Multicenter Pilot AnalysisHydroxycarboxylic acid receptors are essential for breast cancer cells to control their lipid/fatty acid metabolismEffects of pyrazole partial agonists on HCA(2) -mediated flushing and VLDL-triglyceride levels in mice.Medium-chain fatty acid-sensing receptor, GPR84, is a proinflammatory receptorThe role of HCA2 (GPR109A) in regulating macrophage function.Activated niacin receptor HCA2 inhibits chemoattractant-mediated macrophage migration via Gβγ/PKC/ERK1/2 pathway and heterologous receptor desensitization.G-protein-coupled receptor 81 promotes a malignant phenotype in breast cancer through angiogenic factor secretion.Low affinity GPCRs for metabolic intermediates: challenges for pharmacologists.Endogenous metabolites as ligands for G protein-coupled receptors modulating risk factors for metabolic and cardiovascular disease.Trans-cinnamic acid increases adiponectin and the phosphorylation of AMP-activated protein kinase through G-protein-coupled receptor signaling in 3T3-L1 adipocytes.The lactate receptor, G-protein-coupled receptor 81/hydroxycarboxylic acid receptor 1: Expression and action in brain.Cell-surface G-protein-coupled receptors for tumor-associated metabolites: A direct link to mitochondrial dysfunction in cancer.Chemically engineering ligand selectivity at the free fatty acid receptor 2 based on pharmacological variation between species orthologs.Discovery of SCH 900271, a Potent Nicotinic Acid Receptor Agonist for the Treatment of Dyslipidemia.Nicotinic acid increases adiponectin secretion from differentiated bovine preadipocytes through G-protein coupled receptor signaling.Hydroxycarboxylic acid-binding receptorsSupplementing obese Zucker rats with niacin induces the transition of glycolytic to oxidative skeletal muscle fibers.G protein-coupled receptors not currently in the spotlight: free fatty acid receptor 2 and GPR35.Palmitate induces fat accumulation by activating C/EBPβ-mediated G0S2 expression in HepG2 cells.Expression of orphan receptors GPR22 and GPR162 in streptozotocin-induced diabetic rats.The Nuclear Orphan Receptor Nur77 Alleviates Palmitate-induced Fat Accumulation by Down-regulating G0S2 in HepG2 Cells.A two-state model for the kinetics of competitive radioligand binding.Potential Synergies of β-Hydroxybutyrate and Butyrate on the Modulation of Metabolism, Inflammation, Cognition, and General Health.
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P2860
International Union of Basic and Clinical Pharmacology. LXXXII: Nomenclature and Classification of Hydroxy-carboxylic Acid Receptors (GPR81, GPR109A, and GPR109B).
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2011 nî lūn-bûn
@nan
2011 թուականի Մարտին հրատարակուած գիտական յօդուած
@hyw
2011 թվականի մարտին հրատարակված գիտական հոդված
@hy
2011年の論文
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2011年論文
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2011年論文
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2011年論文
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2011年論文
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2011年論文
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2011年论文
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name
International Union of Basic a ...... (GPR81, GPR109A, and GPR109B).
@ast
International Union of Basic a ...... (GPR81, GPR109A, and GPR109B).
@en
International Union of Basic a ...... (GPR81, GPR109A, and GPR109B).
@nl
type
label
International Union of Basic a ...... (GPR81, GPR109A, and GPR109B).
@ast
International Union of Basic a ...... (GPR81, GPR109A, and GPR109B).
@en
International Union of Basic a ...... (GPR81, GPR109A, and GPR109B).
@nl
prefLabel
International Union of Basic a ...... (GPR81, GPR109A, and GPR109B).
@ast
International Union of Basic a ...... (GPR81, GPR109A, and GPR109B).
@en
International Union of Basic a ...... (GPR81, GPR109A, and GPR109B).
@nl
P2093
P356
P1476
International Union of Basic a ...... (GPR81, GPR109A, and GPR109B).
@en
P2093
Graeme Semple
Steven L Colletti
Timothy W Lovenberg
P304
P356
10.1124/PR.110.003301
P577
2011-03-31T00:00:00Z