5-Methyl-1-(3-pyridylcarbamoyl)-1,2,3,5-tetrahydropyrrolo[2,3-f]indole: a novel 5-HT2C/5-HT2B receptor antagonist with improved affinity, selectivity, and oral activity.
about
Head-twitch response in rodents induced by the hallucinogen 2,5-dimethoxy-4-iodoamphetamine: a comprehensive history, a re-evaluation of mechanisms, and its utility as a model.In vitro and in vivo profile of SB 206553, a potent 5-HT2C/5-HT2B receptor antagonist with anxiolytic-like propertiesSimilarities between the Binding Sites of SB-206553 at Serotonin Type 2 and Alpha7 Acetylcholine Nicotinic Receptors: Rationale for Its Polypharmacological ProfilePredicted structures and dynamics for agonists and antagonists bound to serotonin 5-HT2B and 5-HT2C receptors.Expression of serotonin receptors in bone.Regioselective alkylation of 1,3,4,5-tetrahydrobenzo[d]azepin-2-one and biological evaluation of the resulting alkylated products as potentially selective [Formula: see text] agonists.
P2860
5-Methyl-1-(3-pyridylcarbamoyl)-1,2,3,5-tetrahydropyrrolo[2,3-f]indole: a novel 5-HT2C/5-HT2B receptor antagonist with improved affinity, selectivity, and oral activity.
description
1995 nî lūn-bûn
@nan
1995 թուականի Յուլիսին հրատարակուած գիտական յօդուած
@hyw
1995 թվականի հուլիսին հրատարակված գիտական հոդված
@hy
1995年の論文
@ja
1995年論文
@yue
1995年論文
@zh-hant
1995年論文
@zh-hk
1995年論文
@zh-mo
1995年論文
@zh-tw
1995年论文
@wuu
name
5-Methyl-1-(3-pyridylcarbamoyl ...... electivity, and oral activity.
@ast
5-Methyl-1-(3-pyridylcarbamoyl ...... electivity, and oral activity.
@en
5-Methyl-1-(3-pyridylcarbamoyl ...... electivity, and oral activity.
@nl
type
label
5-Methyl-1-(3-pyridylcarbamoyl ...... electivity, and oral activity.
@ast
5-Methyl-1-(3-pyridylcarbamoyl ...... electivity, and oral activity.
@en
5-Methyl-1-(3-pyridylcarbamoyl ...... electivity, and oral activity.
@nl
prefLabel
5-Methyl-1-(3-pyridylcarbamoyl ...... electivity, and oral activity.
@ast
5-Methyl-1-(3-pyridylcarbamoyl ...... electivity, and oral activity.
@en
5-Methyl-1-(3-pyridylcarbamoyl ...... electivity, and oral activity.
@nl
P2093
P356
P1476
5-Methyl-1-(3-pyridylcarbamoyl ...... electivity, and oral activity.
@en
P2093
Blackburn TP
Kennett GA
Thompson M
P304
P356
10.1021/JM00014A004
P407
P577
1995-07-01T00:00:00Z