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Structure-based design of estrogen receptor-beta selective ligands.

Structure-based design of estrogen receptor-beta selective ligands.

http://www.wikidata.org/entity/Q34368597

about

3D models of MBP, a biologically active metabolite of bisphenol A, in human estrogen receptor α and estrogen receptor β Estrogen receptor beta-selective agonists stimulate calcium oscillations in human and mouse embryonic stem cell-derived neurons Confidence limits, error bars and method comparison in molecular modeling. Part 1: the calculation of confidence intervals Regulation of specific target genes and biological responses by estrogen receptor subtype agonists Identification of xenoestrogens in food additives by an integrated in silico and in vitro approach Aerobic Iron-Based Cross-Dehydrogenative Coupling Enables Efficient Diversity-Oriented Synthesis of Coumestrol-Based Selective Estrogen Receptor Modulators Structural overview of the nuclear receptor superfamily: insights into physiology and therapeutics.Identification of ligands with bicyclic scaffolds provides insights into mechanisms of estrogen receptor subtype selectivity.Characterization of the oestrogenic activity of non-aromatic steroids: are there male-specific endogenous oestrogen receptor modulators?Genome-wide dynamics of chromatin binding of estrogen receptors alpha and beta: mutual restriction and competitive site selection.Specific activation of estrogen receptor alpha and beta enhances male sexual behavior and neuroplasticity in male Japanese quail.Targeting estrogen receptor-β for the prevention of nonmelanoma skin cancer.Estrogen receptor beta selective nonsteroidal estrogens: seeking clinical indications.Bisphenol AF is a full agonist for the estrogen receptor ERalpha but a highly specific antagonist for ERbeta Selective ligands of estrogen receptor β discovered using pharmacophore mapping and structure-based virtual screening.Versatility or promiscuity: the estrogen receptors, control of ligand selectivity and an update on subtype selective ligands.Selectively targeting estrogen receptors for cancer treatment.Treatment with an orally bioavailable prodrug of 17β-estradiol alleviates hot flushes without hormonal effects in the periphery.A screening cascade to identify ERβ ligands.Characterization of the estradiol-binding site structure of human pancreas-specific protein disulfide isomerase: indispensable role of the hydrogen bond between His278 and the estradiol 3-hydroxyl group The unexpected science of estrogen receptor-beta selective agonists: a new class of anti-inflammatory agents?Structural characterization of the binding interactions of various endogenous estrogen metabolites with human estrogen receptor α and β subtypes: a molecular modeling study.Estrogen receptor β ligands: recent advances and biomedical applications.Multiple-targeting and conformational selection in the estrogen receptor: computation and experiment.A molecular docking study of phytochemical estrogen mimics from dietary herbal supplements Structural and Functional Diversity of Estrogen Receptor Ligands.Estrogen Receptor β Activation Rapidly Modulates Male Sexual Motivation through the Transactivation of Metabotropic Glutamate Receptor 1a.Bioactivation of Selective Estrogen Receptor Modulators (SERMs)Linkage effects on binding affinity and activation of GPR30 and estrogen receptors ERalpha/beta with tridentate pyridin-2-yl hydrazine tricarbonyl-Re/(99m)Tc(I) chelates.Understanding nuclear receptor form and function using structural biology A medicinal chemist's guide to molecular interactions Role of pocket flexibility in the modulation of estrogen receptor alpha by key residue arginine 394.One-step synthesis of azole- and benzazole-based sulfonamides in aqueous media.

P2860

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P2860

Structure-based design of estrogen receptor-beta selective ligands.

http://www.wikidata.org/entity/Q34368597

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2004 nî lūn-bûn

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2004 թուականի Նոյեմբերին հրատարակուած գիտական յօդուած

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2004 թվականի նոյեմբերին հրատարակված գիտական հոդված

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2004年の論文

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2004年論文

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2004年论文

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name

Structure-based design of estrogen receptor-beta selective ligands.

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Structure-based design of estrogen receptor-beta selective ligands.

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Structure-based design of estrogen receptor-beta selective ligands.

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Structure-based design of estrogen receptor-beta selective ligands.

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Structure-based design of estrogen receptor-beta selective ligands.

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Structure-based design of estrogen receptor-beta selective ligands.

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Structure-based design of estrogen receptor-beta selective ligands.

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Structure-based design of estrogen receptor-beta selective ligands.

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Structure-based design of estrogen receptor-beta selective ligands.

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Journal of the American Chemical Society

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Structure-based design of estrogen receptor-beta selective ligands.

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Ashok Bapat

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Chris P Miller

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Chulai Hsiao

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Eric S Manas

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Heather A Harris

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Juan C Alvarez

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Karl Malakian

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Mark L Stahl

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Michael S Malamas

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Ramesh A Bhat

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scholarly article

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10.1021/JA047633O

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15548008

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