Inhibition of cancer-associated mutant isocitrate dehydrogenases: synthesis, structure-activity relationship, and selective antitumor activity.
about
Targeting histone methylation for cancer therapy: enzymes, inhibitors, biological activity and perspectivesIsocitrate dehydrogenase mutations: new opportunities for translational researchInhibition of Cancer-Associated Mutant Isocitrate Dehydrogenases by 2-Thiohydantoin Compounds3-(Piperidin-4-ylmethoxy)pyridine Containing Compounds Are Potent Inhibitors of Lysine Specific Demethylase 1.Structure based discovery of clomifene as a potent inhibitor of cancer-associated mutant IDH1.Allosteric inhibitor remotely modulates the conformation of the orthestric pockets in mutant IDH2/R140Q.Discovery and Evaluation of Clinical Candidate IDH305, a Brain Penetrant Mutant IDH1 Inhibitor.Optimization of 3-Pyrimidin-4-yl-oxazolidin-2-ones as Allosteric and Mutant Specific Inhibitors of IDH1.Beyond Brooding on Oncometabolic Havoc in IDH-Mutant Gliomas and AML: Current and Future Therapeutic Strategies.2-Hydroxypyridine-N-oxide-Embedded Aurones as Potent Human Tyrosinase Inhibitors.Inhibition of Glycolysis and Glutaminolysis: Emerging Drug Discovery Approach to Combat Cancer.
P2860
Q26744441-18586DA8-28FC-4C53-A557-20D186061FFCQ27001014-4BC15970-8159-40BD-9CE6-DCAE4655E325Q36052714-7AF15F09-2480-4639-89FC-B68BD10A0BB3Q36930863-879E5F55-CCD5-4B23-9413-CC8B0E0C5155Q41279919-68DB21D4-5EF9-4CDE-BCC8-1DAA1F509015Q47139135-8A0EE802-335E-472D-8BD4-915837AB81A1Q48007877-3BD9C957-2CC5-46B4-ACD3-C07F9976C74FQ48308884-21E86700-68A9-433F-A067-66BD0B5DCCE7Q50033966-A21E3670-04C5-4D54-836B-BDB08965E67EQ50333141-53221210-E51B-4F0F-BFBA-D6C39F9D5B5BQ54978523-397A0CF1-3A29-42A4-86B7-4F5DFD06E44A
P2860
Inhibition of cancer-associated mutant isocitrate dehydrogenases: synthesis, structure-activity relationship, and selective antitumor activity.
description
2014 nî lūn-bûn
@nan
2014 թուականի Հոկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2014 թվականի հոտեմբերին հրատարակված գիտական հոդված
@hy
2014年の論文
@ja
2014年論文
@yue
2014年論文
@zh-hant
2014年論文
@zh-hk
2014年論文
@zh-mo
2014年論文
@zh-tw
2014年论文
@wuu
name
Inhibition of cancer-associate ...... selective antitumor activity.
@ast
Inhibition of cancer-associate ...... selective antitumor activity.
@en
Inhibition of cancer-associate ...... selective antitumor activity.
@nl
type
label
Inhibition of cancer-associate ...... selective antitumor activity.
@ast
Inhibition of cancer-associate ...... selective antitumor activity.
@en
Inhibition of cancer-associate ...... selective antitumor activity.
@nl
prefLabel
Inhibition of cancer-associate ...... selective antitumor activity.
@ast
Inhibition of cancer-associate ...... selective antitumor activity.
@en
Inhibition of cancer-associate ...... selective antitumor activity.
@nl
P2093
P2860
P356
P1476
Inhibition of cancer-associate ...... selective antitumor activity.
@en
P2093
Baisong Zheng
James M Gallo
Jihui J Qiu
Lisheng Deng
Mari Kogiso
Xiao-Nan Li
Yongcheng Song
P2860
P304
P356
10.1021/JM500660F
P407
P577
2014-10-01T00:00:00Z