Synthesis and biological activity of a novel series of nonsteroidal, peripherally selective androgen receptor antagonists derived from 1,2-dihydropyridono[5,6-g]quinolines.
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Pharmacokinetics and pharmacodynamics of nonsteroidal androgen receptor ligandsChemistry and structural biology of androgen receptor2-Anilino-3-benzoyl-4-(2,5-dichloro-phen-yl)-7,7-dimethyl-5-oxo-5,6,7,8-tetra-hydro-4H-benzo[b]pyranStructural basis for computational screening of non-steroidal androgen receptor ligands.Male hormonal contraceptives.Dimethyl 2,6,8-trimethyl-1,2-dihydroquinoline-2,4-dicarboxylateAdvances in male hormonal contraception.Dimethyl 2-methyl-1,2-dihydro-quinoline-2,4-dicarboxyl-ate.Dimethyl 6-acetyl-2-methyl-1,2-dihydroquinoline-2,4-dicarboxyl-ate.Dimethyl 6-bromo-2-methyl-1,2-di-hydro-quinoline-2,4-dicarboxyl-ateMolecular targets of androgen signaling that characterize skeletal muscle recovery and regeneration.In vitro and in vivo structure-activity relationships of novel androgen receptor ligands with multiple substituents in the B-ringStructure of the ligand-binding domain (LBD) of human androgen receptor in complex with a selective modulator LGD2226Photocytotoxicity of the fluorescent nonsteroidal androgen receptor ligand TDPQ.Androgen receptor-mediated apoptosis is regulated by photoactivatable androgen receptor ligands.Differential presentation of protein interaction surfaces on the androgen receptor defines the pharmacological actions of bound ligands.Novel and efficient one-step parallel synthesis of dibenzopyranones via Suzuki-Miyaura cross coupling.Potent, nonsteroidal selective androgen receptor modulators (SARMs) based on 8H-[1,4]oxazino[2,3-f]quinolin-8-ones.A Copper-Catalyzed Tandem Cyclization Reaction of Aminoalkynes with Alkynes for the Construction of Tetrahydropyrrolo[1,2-a]quinolines Scaffold.Synthesis and pharmacological evaluation of dimeric follicle-stimulating hormone receptor antagonists.Recent discoveries and developments of androgen receptor based therapy for prostate cancerDiscovery and Identification of Pyrazolopyramidine Analogs as Novel Potent Androgen Receptor Antagonists
P2860
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P2860
Synthesis and biological activity of a novel series of nonsteroidal, peripherally selective androgen receptor antagonists derived from 1,2-dihydropyridono[5,6-g]quinolines.
description
1998 nî lūn-bûn
@nan
1998 թուականի Փետրուարին հրատարակուած գիտական յօդուած
@hyw
1998 թվականի փետրվարին հրատարակված գիտական հոդված
@hy
1998年の論文
@ja
1998年論文
@yue
1998年論文
@zh-hant
1998年論文
@zh-hk
1998年論文
@zh-mo
1998年論文
@zh-tw
1998年论文
@wuu
name
Synthesis and biological activ ...... ydropyridono[5,6-g]quinolines.
@ast
Synthesis and biological activ ...... ydropyridono[5,6-g]quinolines.
@en
Synthesis and biological activ ...... ydropyridono[5,6-g]quinolines.
@nl
type
label
Synthesis and biological activ ...... ydropyridono[5,6-g]quinolines.
@ast
Synthesis and biological activ ...... ydropyridono[5,6-g]quinolines.
@en
Synthesis and biological activ ...... ydropyridono[5,6-g]quinolines.
@nl
prefLabel
Synthesis and biological activ ...... ydropyridono[5,6-g]quinolines.
@ast
Synthesis and biological activ ...... ydropyridono[5,6-g]quinolines.
@en
Synthesis and biological activ ...... ydropyridono[5,6-g]quinolines.
@nl
P2093
P356
P1476
Synthesis and biological activ ...... ydropyridono[5,6-g]quinolines.
@en
P2093
Edwards JP
Higuchi RI
Marschke KB
P304
P356
10.1021/JM970699S
P407
P577
1998-02-01T00:00:00Z